PDB-code
Browse kinase entries (page 128 of 282)
First 124 125 126 PreviousLast132 131 130 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | GAK | NAK | Other | 4c58 | A | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show |  |
| GAK | NAK | Other | 4c59 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4c59 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4o38 | A | A | - | Human | Show | |
| GAK | NAK | Other | 4o38 | A | B | - | Human | Show | |
| GAK | NAK | Other | 4o38 | B | A | - | Human | Show | |
| GAK | NAK | Other | 4o38 | B | B | - | Human | Show | |
| GAK | NAK | Other | 4y8d | A | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | Show | |
| GAK | NAK | Other | 4y8d | A | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | Show | |
| GAK | NAK | Other | 4y8d | B | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | Show | |
| GAK | NAK | Other | 4y8d | B | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | Show | |
| GAK | NAK | Other | 5y7z | A | gefitinib | Human | Show | | |
| GAK | NAK | Other | 5y7z | B | gefitinib | Human | Show | | |
| GAK | NAK | Other | 5y80 | A | A | gefitinib | Human | Show | |
| GAK | NAK | Other | 5y80 | A | B | gefitinib | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 3cik | A | - | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 3krw | A | balanol | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 3krx | A | balanol | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | A | paroxetine | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | B | paroxetine | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | A | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | B | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | A | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | B | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | A | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | B | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | A | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | B | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | A | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | B | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5uvc | A | n-benzyl-3-({[5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)benzamide | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 5wg3 | A | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamide | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | A | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | B | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 6c2y | A | (4r,5r,6s)-4-[4-fluoro-3-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)phenyl]-n-(2h-indazol-5-yl)-6-methyl-2-oxohexahydropyrimidine-5-carboxamide | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 6u7c | A | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(2h-indazol-3-yl)methyl]benzamide | Human | Show | | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | A | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | B | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | A | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | B | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | A | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | Show | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | B | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | Show | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | A | amp phosphoramidate | Human | Show | | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | B | amp phosphoramidate | Human | Show | | |
| GRK5 (GPRK5) | GRK | AGC | 4tnb | A | sangivamycin | Human | Show | | |
| GRK5 (GPRK5) | GRK | AGC | 4tnd | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
