PDB-code
Browse kinase entries (page 168 of 282)
First 164 165 166 PreviousLast172 171 170 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | A | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | A | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | B | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | B | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 7szr | A | A | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 7szr | A | B | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4dn5 | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4dn5 | B | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4g3d | A | - | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4g3d | B | - | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4g3d | D | - | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4g3d | E | - | Human | Show | ![]() | |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idt | A | A | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idt | A | B | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idt | B | A | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idt | B | B | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idv | A | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idv | B | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idv | C | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 4idv | D | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6wpp | A | A | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6wpp | A | B | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6wpp | B | A | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6wpp | B | B | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1q | A | A | desf-3r/4076 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1q | A | B | desf-3r/4076 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1q | B | A | desf-3r/4076 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1q | B | B | desf-3r/4076 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1t | A | A | 4s/3694 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1t | A | B | 4s/3694 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1t | B | A | 4s/3694 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 6z1t | B | B | 4s/3694 | Human | Show | ![]() |
![]() | MAP3K14 (NIK) | STE-Unique | STE | 8yhw | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5hes | A | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5hes | A | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5hes | B | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5hes | B | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | A | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | B | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 6jut | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]-3-bromanyl-benzenesulfonamide | Human | Show | ![]() |


