PDB-code
Browse kinase entries (page 171 of 282)
First 167 168 169 PreviousLast175 174 173 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAP3K7 (TAK1) | MLK | TKL | 5j8i | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | Show |  | |
| MAP3K7 (TAK1) | MLK | TKL | 5j9l | A | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5jga | A | n-[5-(4-methylpiperazine-1-carbonyl)[1,1'-biphenyl]-2-yl]-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgb | A | n-(2-methoxy-4-{[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgd | A | n-(2-isopropoxy-3-(4-methylpiperazine-1-carbonyl)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5jh6 | A | 2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl prop-2-enoate | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5jk3 | A | ~{n}-[2-[5-chloranyl-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | A | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | B | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | A | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | B | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | A | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | B | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 8gw3 | A | - | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | A | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | B | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | C | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | A | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | B | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | C | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | |
| MAP3K9 (MLK1) | MLK | TKL | 3dtc | A | 12-(2-hydroxyethyl)-2-(1-methylethoxy)-13,14-dihydronaphtho[2,1-a]pyrrolo[3,4-c]carbazol-5(12h)-one | Human | Show | | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | A | - | Human | Show | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | B | - | Human | Show | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | A | - | Human | Show | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | B | - | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqd | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqd | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | A | A | - | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | A | B | - | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | B | A | - | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | B | B | - | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqf | A | n-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amine | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | B | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | B | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfz | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfz | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6ng0 | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 6ng0 | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 7kac | A | 5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-one | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 7kac | B | 5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-one | Human | Show | | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | A | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | A | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | B | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | Show | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | B | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | Show | |
