PDB-code
Browse kinase entries (page 177 of 282)
First 173 174 175 PreviousLast181 180 179 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | Show |  |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | A | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | B | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | A | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | B | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | A | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | B | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | A | - | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | B | - | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opg | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 6oph | A | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opi | A | (3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamide | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7k | A | 1h-imidazol-2-amine | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | A | - | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | B | - | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | A | 1,2-oxazol-3-amine | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | B | 1,2-oxazol-3-amine | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | A | pyridin-2-amine | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | B | pyridin-2-amine | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | A | pyrazole | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | B | pyrazole | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | A | 1~{h}-pyridin-2-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | B | 1~{h}-pyridin-2-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | A | 1~{h}-1,2,3-triazole | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | B | 1~{h}-1,2,3-triazole | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | A | 1-azanylpropylideneazanium | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | B | 1-azanylpropylideneazanium | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | A | 1,1-bis(oxidanylidene)thietan-3-ol | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | B | 1,1-bis(oxidanylidene)thietan-3-ol | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | A | thiophen-3-ylmethylazanium | Human | Show | |
