PDB-code
Browse kinase entries (page 178 of 282)
First 174 175 176 PreviousLast182 181 180 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | B | thiophen-3-ylmethylazanium | Human | Show |  |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | A | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | B | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rfo | A | - | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | A | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | B | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | A | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | B | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e73 | A | - | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e75 | A | - | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | A | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | B | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | A | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | B | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7w5o | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 7xc1 | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | A | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | B | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | A | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | B | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | A | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | B | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | A | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | B | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | A | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | B | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | C | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | A | ~{n}-pyridin-3-ylprop-2-enamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | B | ~{n}-pyridin-3-ylpropanamide | Human | Show | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | A | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | Show | |
