PDB-code
Browse kinase entries (page 190 of 282)
First 186 187 188 PreviousLast194 193 192 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK14 (p38a) | MAPK | CMGC | 3iw5 | A | n-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamide | Human | Show |  | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | A | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | B | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw7 | A | 2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw8 | A | 1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | A | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | B | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3j | A | 2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3kf7 | A | 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | A | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | B | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8s | A | 3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8x | A | n,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfa | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfc | A | (4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfd | A | 1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfe | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | A | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | B | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lhj | A | n-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mgy | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh0 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh1 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh2 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh3 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpa | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | A | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | B | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | A | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | B | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | A | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | B | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mw1 | A | 8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | A | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | B | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | A | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | B | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | B | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnx | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3nww | A | 1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylurea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8p | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8t | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8u | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3obg | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3obj | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | |
