PDB-code
Browse kinase entries (page 216 of 282)
First 212 213 214 PreviousLast220 219 218 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | A | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | B | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2pe0 | A | 5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-one | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2pe1 | A | 1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}urea | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2pe2 | A | 3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamide | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2r7b | A | 10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamine | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2xch | A | 8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 2xck | A | 1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3h9o | A | 2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amine | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | A | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | B | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | A | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | B | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3ion | A | 2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3iop | A | 2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nax | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nay | A | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nay | B | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | A | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | B | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | A | 1h-indazol-3-amine | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | B | 1h-indazol-3-amine | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | A | 3,4-dihydroisoquinolin-1(2h)-one | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | B | 3,4-dihydroisoquinolin-1(2h)-one | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | A | quinazolin-4(1h)-one | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | B | quinazolin-4(1h)-one | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | A | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | B | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | C | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | D | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | E | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | F | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | G | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orx | H | - | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3otu | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3pwy | A | n-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamide | Human | Show | ![]() | |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | A | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | B | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | Show | ![]() |


