Browse kinase entries (page 216 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PDPK1 (PDK1)PDK1AGC2biyAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC2biyABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC2pe0A5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-oneHumanShow
PDPK1 (PDK1)PDK1AGC2pe1A1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}ureaHumanShow
PDPK1 (PDK1)PDK1AGC2pe2A3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamideHumanShow
PDPK1 (PDK1)PDK1AGC2r7bA10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamineHumanShow
PDPK1 (PDK1)PDK1AGC2xchA8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC2xckA1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3h9oA2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amineHumanShow
PDPK1 (PDK1)PDK1AGC3hrcAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC3hrcABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC3hrfAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC3hrfABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC3ionA2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHumanShow
PDPK1 (PDK1)PDK1AGC3iopA2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHumanShow
PDPK1 (PDK1)PDK1AGC3naxA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3nayA4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3nayB4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3nunAA6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3nunAB6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3nusAA1h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3nusAB1h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3nuuAA3,4-dihydroisoquinolin-1(2h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3nuuAB3,4-dihydroisoquinolin-1(2h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3nuyAAquinazolin-4(1h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3nuyABquinazolin-4(1h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC3orxA-HumanShow
PDPK1 (PDK1)PDK1AGC3orxB-HumanShow
PDPK1 (PDK1)PDK1AGC3orxC-HumanShow
PDPK1 (PDK1)PDK1AGC3orxD-HumanShow
PDPK1 (PDK1)PDK1AGC3orxE-HumanShow
PDPK1 (PDK1)PDK1AGC3orxF-HumanShow
PDPK1 (PDK1)PDK1AGC3orxG-HumanShow
PDPK1 (PDK1)PDK1AGC3orxH-HumanShow
PDPK1 (PDK1)PDK1AGC3orzAA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzAB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzBA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzBB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzCA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzCB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzDA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3orzDB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3otuA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC3pwyAn-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamideHumanShow
PDPK1 (PDK1)PDK1AGC3qc4AA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qc4AB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qc4BA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qc4BB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qcqAA6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHumanShow
PDPK1 (PDK1)PDK1AGC3qcqAB6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHumanShow
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