Version: 3.2
Updated: 01-Nov-2025

Browse kinase entries (page 225 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
Pik3cd (p110d)PIKAtypical7porA~{n}-[2-[2-fluoranyl-4-[(4-propan-2-ylpiperazin-1-yl)methyl]phenyl]pyridin-4-yl]-2-methoxy-5-morpholin-4-yl-pyridine-3-sulfonamideMouseShow
Pik3cd (p110d)PIKAtypical7posA5-(3,6-dihydro-2~{h}-pyran-4-yl)-2-methoxy-~{n}-[5-[3-(4-propan-2-ylpiperazin-1-yl)prop-1-ynyl]pyridin-3-yl]pyridine-3-sulfonamideMouseShow
Pik3cd (p110d)PIKAtypical7potAn-[5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxy-pyridin-3-yl]benzenesulfonamideMouseShow
Pik3cd (p110d)PIKAtypical7r26A5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amineMouseShow
Pik3cd (p110d)PIKAtypical7r2bA(4~{s})-3-[6-[2-azanyl-4-(trifluoromethyl)pyrimidin-5-yl]-2-morpholin-4-yl-pyrimidin-4-yl]-4-methyl-1,3-oxazolidin-2-oneMouseShow
PIK3CD (p110d)PIKAtypical5dxuA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHumanShow
PIK3CD (p110d)PIKAtypical5m6uA4-azanyl-6-[[(1~{s})-1-(4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]pyrimidine-5-carbonitrileHumanShow
PIK3CD (p110d)PIKAtypical5t8fA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHumanShow
PIK3CD (p110d)PIKAtypical5ubtA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHumanShow
PIK3CD (p110d)PIKAtypical5vlrA4-acetyl-1-(3-{4-amino-5-[1-(2,2,2-trifluoroethyl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)-3,3-dimethylpiperazin-2-oneHumanShow
PIK3CD (p110d)PIKAtypical6g6wAA~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHumanShow
PIK3CD (p110d)PIKAtypical6g6wAB~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHumanShow
PIK3CD (p110d)PIKAtypical6ocoA4-[(1s,4s)-5-(3-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carbonitrileHumanShow
PIK3CD (p110d)PIKAtypical6ocuA5-{(3r)-3-methyl-4-[(1r,2r)-2-methylcyclopropane-1-carbonyl]piperazin-1-yl}-3-(1-methyl-1h-pyrazol-4-yl)pyrazine-2-carbonitrileHumanShow
PIK3CD (p110d)PIKAtypical6pyrAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHumanShow
PIK3CD (p110d)PIKAtypical6pyrAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHumanShow
PIK3CD (p110d)PIKAtypical6pyuA(3s)-1'-(cyclopropanecarbonyl)-5-(quinoxalin-6-yl)spiro[indole-3,2'-pyrrolidin]-2(1h)-oneHumanShow
PIK3CD (p110d)PIKAtypical7jisA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHumanShow
PIK3CD (p110d)PIKAtypical7lm2Acyclopropyl[(3s)-3-{[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]amino}pyrrolidin-1-yl]methanoneHumanShow
PIK3CD (p110d)PIKAtypical7lq1An-(5-(6-(2-((2s,6r)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamideHumanShow
PIK3CD (p110d)PIKAtypical8bcyAA9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHumanShow
PIK3CD (p110d)PIKAtypical8bcyAB9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHumanShow
PIK3CG (p110g)PIKAtypical1e8yA-HumanShow
PIK3CG (p110g)PIKAtypical1e8zAstaurosporineHumanShow
PIK3CG (p110g)PIKAtypical1he8A-HumanShow
PIK3CG (p110g)PIKAtypical2a4zA(5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dioneHumanShow
PIK3CG (p110g)PIKAtypical2a5uA(5e)-5-(quinoxalin-6-ylmethylene)-1,3-thiazolidine-2,4-dioneHumanShow
PIK3CG (p110g)PIKAtypical2chwA2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-oneHumanShow
PIK3CG (p110g)PIKAtypical2chxAn-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamideHumanShow
PIK3CG (p110g)PIKAtypical2chzAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PIK3CG (p110g)PIKAtypical2v4lA3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenolHumanShow
PIK3CG (p110g)PIKAtypical3apcA5-(7-methanesulfonyl-2-morpholin-4-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHumanShow
PIK3CG (p110g)PIKAtypical3apdA5-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHumanShow
PIK3CG (p110g)PIKAtypical3apfA3-[7-(1h-benzimidazol-5-yl)-2-(morpholin-4-yl)-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl]phenolHumanShow
PIK3CG (p110g)PIKAtypical3csfA-HumanShow
PIK3CG (p110g)PIKAtypical3cstAmethylated ruthenium pyridocarbazoleHumanShow
PIK3CG (p110g)PIKAtypical3dbsA2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidineHumanShow
PIK3CG (p110g)PIKAtypical3dpdA5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-oneHumanShow
PIK3CG (p110g)PIKAtypical3eneA1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amineHumanShow
PIK3CG (p110g)PIKAtypical3ibeA1-(4-{4-morpholin-4-yl-1-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-6-yl}phenyl)-3-pyridin-4-ylureaHumanShow
PIK3CG (p110g)PIKAtypical3l08AA2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHumanShow
PIK3CG (p110g)PIKAtypical3l08AB2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHumanShow
PIK3CG (p110g)PIKAtypical3l13A[3-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenyl]methanolHumanShow
PIK3CG (p110g)PIKAtypical3l16A5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyridin-2-amineHumanShow
PIK3CG (p110g)PIKAtypical3l17A4-methyl-5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyrimidin-2-amineHumanShow
PIK3CG (p110g)PIKAtypical3l54A6-(1h-pyrazolo[3,4-b]pyridin-5-yl)-4-pyridin-4-ylquinolineHumanShow
PIK3CG (p110g)PIKAtypical3lj3A(2z)-4,6-dihydroxy-2-{[1-methyl-4-(4-methylpiperazin-1-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-1-benzofuran-3(2h)-oneHumanShow
PIK3CG (p110g)PIKAtypical3mjwA(2z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2h)-oneHumanShow
PIK3CG (p110g)PIKAtypical3ml8A8-cyclopentyl-6-[3-(hydroxymethyl)phenyl]-4-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
PIK3CG (p110g)PIKAtypical3ml9A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
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