PDB-code
Browse kinase entries (page 227 of 282)
First 223 224 225 PreviousLast231 230 229 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | PIK3CG (p110g) | PIK | Atypical | 4ps8 | A | n-[6-(5,6-dimethoxypyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | Show |  | |
| PIK3CG (p110g) | PIK | Atypical | 4urk | A | 2-[[(1r)-1-(7-methyl-2-morpholin-4-yl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-9-yl)ethyl]amino]benzoic acid | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4wwn | A | n-{(1s)-1-[7-fluoro-2-(pyridin-2-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4wwo | A | n-{(1s)-1-[8-chloro-2-(3-fluorophenyl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4wwp | A | n-{(1s)-1-[8-chloro-2-(2-methylpyridin-3-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4xx5 | A | n-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4xz4 | A | n-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5eds | A | 4-azanyl-6-[[(1~{s})-1-[6-fluoranyl-1-(3-methylsulfonylphenyl)benzimidazol-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5g2n | A | 2-azanyl-~{n}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5g55 | A | 6-cyano-4-[[(1r)-1-(4-methylphenyl)ethyl]amino]quinoline-3-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5jha | A | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)pyrimidin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5jhb | A | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5kae | A | 4-azanyl-6-[[(1~{s})-1-(6-fluoranyl-3-phenyl-4-piperazin-1-ylcarbonyl-quinolin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | A | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | B | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 5t23 | A | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | A | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | B | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 6c1s | A | {4-[2-(5,6-dimethoxypyridin-3-yl)-5-oxo-5,7-dihydro-6h-pyrrolo[3,4-b]pyridin-6-yl]-1h-pyrazol-1-yl}acetonitrile | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6fh5 | A | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6gq7 | A | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6t3b | A | 2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6t3c | A | 7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6xrl | A | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6xrm | A | 5-[2-amino-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1s)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1h-isoindol-1-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 6xrn | A | 2-amino-5-{2-[(1s)-1-cyclopropylethyl]-7-methyl-1-oxo-2,3-dihydro-1h-isoindol-5-yl}-n-(trans-3-hydroxycyclobutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7jwe | A | gedatolisib | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7jwz | A | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7jx0 | A | n~3~-{[5-(4-acetylphenyl)-4-methyl-1,3-thiazol-2-yl]carbamoyl}-n-tert-butyl-beta-alaninamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7kke | A | n-[2-(3,3-dimethylbutoxy)ethyl]-n'-{4-methyl-5-[(pyridin-4-yl)ethynyl]-1,3-thiazol-2-yl}urea | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7mez | A | - | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 7z61 | A | 9-[(3~{r},4~{r})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 8dp0 | A | - | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | A | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | B | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | C | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | Show | |
| PIK3R4 | VPS15 | Other | 7bl1 | C | - | Human | Show | | |
| PIK3R4 | VPS15 | Other | 8sor | D | - | Human | Show | | |
| PIM1 | PIM | CAMK | 1xqz | A | - | Human | Show | | |
| PIM1 | PIM | CAMK | 1xr1 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| PIM1 | PIM | CAMK | 1xws | A | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | Show | |
| PIM1 | PIM | CAMK | 1xws | A | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | Show | |
| PIM1 | PIM | CAMK | 1yhs | A | staurosporine | Human | Show | | |
| PIM1 | PIM | CAMK | 1yi3 | A | 2-morpholin-4-yl-7-phenyl-4h-chromen-4-one | Human | Show | | |
| PIM1 | PIM | CAMK | 1yi4 | A | adenosine | Human | Show | | |
| PIM1 | PIM | CAMK | 1ywv | A | A | - | Human | Show | |
| PIM1 | PIM | CAMK | 1ywv | A | B | - | Human | Show | |
| PIM1 | PIM | CAMK | 1yxs | A | A | - | Human | Show | |
| PIM1 | PIM | CAMK | 1yxs | A | B | - | Human | Show | |
| PIM1 | PIM | CAMK | 1yxt | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
