PDB-code
Browse kinase entries (page 232 of 282)
First 228 229 230 PreviousLast236 235 234 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PIM1 | PIM | CAMK | 5v80 | A | 1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5v82 | A | 1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5vua | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vua | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vub | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vub | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vub | B | C | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vuc | B | A | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5vuc | B | B | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6ayd | A | A | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6ayd | A | B | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6bsk | A | 4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acid | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6kzi | A | 4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l11 | A | 5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l12 | A | 4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l13 | A | 2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l14 | A | 2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l15 | A | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l16 | A | 2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6l17 | A | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6mt0 | A | 3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6no8 | A | 5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6no9 | A | 5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6pcw | A | 4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6pdi | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6pdn | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6pdn | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6pdo | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6pdo | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6pdp | A | A | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6pdp | A | B | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6qxk | B | A | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6qxk | B | B | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6vru | A | A | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6vru | A | B | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6vrv | A | 4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 6ykd | A | A | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 6ykd | A | B | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7oov | A | ~{n}-[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-azanyl-5-[[$l^{1}-azanyl($l^{2}-azanylidene)methyl]-$l^{2}-azanyl]-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]-9-oxidanylidene-9-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]nonanamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 7oow | A | - | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 7oox | A | A | - | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7oox | A | B | - | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7qb2 | A | 4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acid | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 7qfm | A | A | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7qfm | A | B | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7vsy | A | - | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 7xsv | A | A | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7xsv | A | B | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7z6u | A | A | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 7z6u | A | B | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | Show | ![]() |


