Browse kinase entries (page 232 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PIM1PIMCAMK5v80A1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-oneHumanShow
PIM1PIMCAMK5v82A1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridineHumanShow
PIM1PIMCAMK5vuaBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vuaBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vubBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vubBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vubBC(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vucBA(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK5vucBB(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHumanShow
PIM1PIMCAMK6aydAAn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHumanShow
PIM1PIMCAMK6aydABn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHumanShow
PIM1PIMCAMK6bskA4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acidHumanShow
PIM1PIMCAMK6kziA4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amineHumanShow
PIM1PIMCAMK6l11A5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amineHumanShow
PIM1PIMCAMK6l12A4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amineHumanShow
PIM1PIMCAMK6l13A2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazineHumanShow
PIM1PIMCAMK6l14A2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazineHumanShow
PIM1PIMCAMK6l15A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazineHumanShow
PIM1PIMCAMK6l16A2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamineHumanShow
PIM1PIMCAMK6l17A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amineHumanShow
PIM1PIMCAMK6mt0A3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-oneHumanShow
PIM1PIMCAMK6no8A5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHumanShow
PIM1PIMCAMK6no9A5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHumanShow
PIM1PIMCAMK6pcwA4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamideHumanShow
PIM1PIMCAMK6pdiA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PIM1PIMCAMK6pdnAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHumanShow
PIM1PIMCAMK6pdnAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHumanShow
PIM1PIMCAMK6pdoAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHumanShow
PIM1PIMCAMK6pdoAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHumanShow
PIM1PIMCAMK6pdpAA5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHumanShow
PIM1PIMCAMK6pdpAB5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHumanShow
PIM1PIMCAMK6qxkBA2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHumanShow
PIM1PIMCAMK6qxkBB2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHumanShow
PIM1PIMCAMK6vruAA3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHumanShow
PIM1PIMCAMK6vruAB3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHumanShow
PIM1PIMCAMK6vrvA4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHumanShow
PIM1PIMCAMK6ykdAA~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHumanShow
PIM1PIMCAMK6ykdAB~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHumanShow
PIM1PIMCAMK7oovA~{n}-[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-azanyl-5-[[$l^{1}-azanyl($l^{2}-azanylidene)methyl]-$l^{2}-azanyl]-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]-9-oxidanylidene-9-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]nonanamideHumanShow
PIM1PIMCAMK7oowA-HumanShow
PIM1PIMCAMK7ooxAA-HumanShow
PIM1PIMCAMK7ooxAB-HumanShow
PIM1PIMCAMK7qb2A4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acidHumanShow
PIM1PIMCAMK7qfmAA4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHumanShow
PIM1PIMCAMK7qfmAB4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHumanShow
PIM1PIMCAMK7vsyA-HumanShow
PIM1PIMCAMK7xsvAA8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHumanShow
PIM1PIMCAMK7xsvAB8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHumanShow
PIM1PIMCAMK7z6uAA4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHumanShow
PIM1PIMCAMK7z6uAB4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHumanShow
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