Browse kinase entries (page 233 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PIM1PIMCAMK7zunA(4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-olHumanShow
PIM1PIMCAMK8afrAA4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHumanShow
PIM1PIMCAMK8afrAB4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHumanShow
PIM1PIMCAMK8r10AA(z)-4-(4-hydroxystyryl)benzoic acidHumanShow
PIM1PIMCAMK8r10AB(z)-4-(4-hydroxystyryl)benzoic acidHumanShow
PIM1PIMCAMK8r18AA(e)-4-(4-hydroxystyryl)benzoic acidHumanShow
PIM1PIMCAMK8r18AB(e)-4-(4-hydroxystyryl)benzoic acidHumanShow
PIM1PIMCAMK8r1nA4-(4-hydroxyphenethyl)benzoic acidHumanShow
PIM1PIMCAMK8r1pA4-(4-aminostyryl)benzoic acidHumanShow
PIM1PIMCAMK8r1tAA4-(4-aminophenethyl)benzoic acidHumanShow
PIM1PIMCAMK8r1tAB4-(4-aminophenethyl)benzoic acidHumanShow
PIM2PIMCAMK2iwiAruthenium-pyridocarbazole-1HumanShow
PIM2PIMCAMK2iwiBruthenium-pyridocarbazole-1HumanShow
PIM2PIMCAMK4x7qA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHumanShow
PIM2PIMCAMK4x7qB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther3p1aAA-HumanShow
PKMYT1 (MYT1)WEEOther3p1aAB-HumanShow
PKMYT1 (MYT1)WEEOther5vcvAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther5vcwA(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHumanShow
PKMYT1 (MYT1)WEEOther5vcwB(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHumanShow
PKMYT1 (MYT1)WEEOther5vcxAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHumanShow
PKMYT1 (MYT1)WEEOther5vcyAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
PKMYT1 (MYT1)WEEOther5vcyAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
PKMYT1 (MYT1)WEEOther5vczAA4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
PKMYT1 (MYT1)WEEOther5vczAB4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
PKMYT1 (MYT1)WEEOther5vd0A1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
PKMYT1 (MYT1)WEEOther5vd1AAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther5vd1ABn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther5vd3An-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHumanShow
PKMYT1 (MYT1)WEEOther8d6cA(1p)-2-amino-6-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther8d6dA(1p)-2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther8d6eAA(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther8d6eAB(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther8d6fA(1m)-2-amino-1-(5-hydroxy-2-methylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHumanShow
PKMYT1 (MYT1)WEEOther8wjyAA[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHumanShow
PKMYT1 (MYT1)WEEOther8wjyAB[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHumanShow
PKN1PKNAGC4otdAA-HumanShow
PKN1PKNAGC4otdAB-HumanShow
PKN1PKNAGC4otgAAlestaurtinibHumanShow
PKN1PKNAGC4otgABlestaurtinibHumanShow
PKN1PKNAGC4othAA-HumanShow
PKN1PKNAGC4othAB-HumanShow
PKN1PKNAGC4otiAA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHumanShow
PKN1PKNAGC4otiAB3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHumanShow
PKN2PKNAGC4crsAphosphothiophosphoric acid-adenylate esterHumanShow
PLK1PLKOther2ou7AAphosphoaminophosphonic acid-adenylate esterHumanShow
PLK1PLKOther2ou7ABphosphoaminophosphonic acid-adenylate esterHumanShow
PLK1PLKOther2owbAA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
PLK1PLKOther2owbAB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
PLK1PLKOther2rkuAA4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHumanShow
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