PDB-code
Browse kinase entries (page 233 of 282)
First 229 230 231 PreviousLast237 236 235 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PIM1 | PIM | CAMK | 7zun | A | (4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-ol | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 8afr | A | A | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8afr | A | B | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r10 | A | A | (z)-4-(4-hydroxystyryl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r10 | A | B | (z)-4-(4-hydroxystyryl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r18 | A | A | (e)-4-(4-hydroxystyryl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r18 | A | B | (e)-4-(4-hydroxystyryl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r1n | A | 4-(4-hydroxyphenethyl)benzoic acid | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 8r1p | A | 4-(4-aminostyryl)benzoic acid | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 8r1t | A | A | 4-(4-aminophenethyl)benzoic acid | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 8r1t | A | B | 4-(4-aminophenethyl)benzoic acid | Human | Show | ![]() |
![]() | PIM2 | PIM | CAMK | 2iwi | A | ruthenium-pyridocarbazole-1 | Human | Show | ![]() | |
![]() | PIM2 | PIM | CAMK | 2iwi | B | ruthenium-pyridocarbazole-1 | Human | Show | ![]() | |
![]() | PIM2 | PIM | CAMK | 4x7q | A | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | Show | ![]() | |
![]() | PIM2 | PIM | CAMK | 4x7q | B | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 3p1a | A | A | - | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 3p1a | A | B | - | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcv | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcw | A | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcw | B | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcx | A | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcy | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcy | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcz | A | A | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vcz | A | B | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vd0 | A | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vd1 | A | A | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vd1 | A | B | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 5vd3 | A | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 8d6c | A | (1p)-2-amino-6-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 8d6d | A | (1p)-2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 8d6e | A | A | (1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamide | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 8d6e | A | B | (1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamide | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 8d6f | A | (1m)-2-amino-1-(5-hydroxy-2-methylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() | |
![]() | PKMYT1 (MYT1) | WEE | Other | 8wjy | A | A | [6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanone | Human | Show | ![]() |
![]() | PKMYT1 (MYT1) | WEE | Other | 8wjy | A | B | [6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanone | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4otd | A | A | - | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4otd | A | B | - | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4otg | A | A | lestaurtinib | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4otg | A | B | lestaurtinib | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4oth | A | A | - | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4oth | A | B | - | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4oti | A | A | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | Show | ![]() |
![]() | PKN1 | PKN | AGC | 4oti | A | B | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | Show | ![]() |
![]() | PKN2 | PKN | AGC | 4crs | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | PLK1 | PLK | Other | 2ou7 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | PLK1 | PLK | Other | 2ou7 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | PLK1 | PLK | Other | 2owb | A | A | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | Show | ![]() |
![]() | PLK1 | PLK | Other | 2owb | A | B | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | Show | ![]() |
![]() | PLK1 | PLK | Other | 2rku | A | A | 4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | Show | ![]() |


