PDB-code
Browse kinase entries (page 254 of 282)
First 250 251 252 PreviousLast258 257 256 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | A | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | Show |  |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | B | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | Show | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | A | staurosporine | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | B | staurosporine | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a61 | A | staurosporine | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a62 | A | staurosporine | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3we4 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | A | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | B | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | A | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | B | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | A | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | B | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf8 | A | 2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl 7,8,9,10-tetrahydro-6h-cyclohepta[b]quinoline-11-carboxylate | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf9 | A | (2s)-1-oxo-1-[(4-sulfamoylphenyl)amino]propan-2-yl (2s)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3j | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3l | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l42 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l43 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l44 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l45 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l46 | A | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | A | [(amino-kappan)methanethiolato](3-fluoro-9-hydroxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | B | staurosporine | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlp | A | [(amino-kappan)methanethiolato](3-fluoro-9-methoxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(n-methyl-1,4,7-trithiecan-9-amine-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n91 | A | 4-{[(1s)-1-(3-fluorophenyl)-2-(methylamino)ethyl]amino}quinazoline-8-carboxamide | Human | Show | | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | A | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | Show | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | B | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | Show | |
| RYK | Ryk | TK | 6tua | A | - | Human | Show | | |
| SGK1 | SGK | AGC | 2r5t | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| SGK1 | SGK | AGC | 3hdm | A | 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | Show | | |
| SGK1 | SGK | AGC | 3hdn | A | [4-(5-naphthalen-2-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)phenyl]acetic acid | Human | Show | | |
| SGK1 | SGK | AGC | 7pue | A | 6-[4-[[2,3-bis(chloranyl)phenyl]sulfonylamino]phenyl]-~{n}-[(3~{r})-pyrrolidin-3-yl]-2~{h}-pyrazolo[3,4-b]pyridine-4-carboxamide | Human | Show | | |
| SIK3 (QSK) | CAMKL | CAMK | 8oku | A | ~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamide | Human | Show | | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4o | A | 2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamide | Human | Show | | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4q | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4u | A | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4v | A | 1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]urea | Human | Show | | |
| SLK | STE20 | STE | 2j51 | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | | |
| SLK | STE20 | STE | 2jfl | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | | |
| SLK | STE20 | STE | 2jfm | A | A | - | Human | Show | |
| SLK | STE20 | STE | 2jfm | A | B | - | Human | Show | |
| SLK | STE20 | STE | 2uv2 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | Show | |
| SLK | STE20 | STE | 2uv2 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | Show | |
