PDB-code
Browse kinase entries (page 259 of 282)
First 255 256 257 PreviousLast263 262 261 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | STK24 (MST3) | STE20 | STE | 4qmn | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show |  |
| STK24 (MST3) | STE20 | STE | 4qmn | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | A | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | B | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmp | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | A | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | B | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qms | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qms | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmt | A | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmv | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| STK24 (MST3) | STE20 | STE | 4qmx | A | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qmy | A | staurosporine | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qmz | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qna | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qo9 | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4qo9 | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4u8z | A | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4w8d | A | 5-(1-methyl-1h-pyrazol-4-yl)-4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidine | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 4w8e | A | 3-{4-[(2r)-2-(5-methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b30 | A | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | A | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | B | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 7b32 | A | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[(2-methoxyphenyl)amino]pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b33 | A | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[4-[6-[bis(fluoranyl)methyl]pyridin-2-yl]-2-chloranyl-phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b34 | A | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranyl-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b35 | A | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 7b35 | B | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | A | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | B | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | A | macrocyclic inhibitor | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | B | macrocyclic inhibitor | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qlr | A | 8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| STK24 (MST3) | STE20 | STE | 8qls | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qls | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qls | A | C | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| STK25 (YSK1) | STE20 | STE | 2xik | A | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| STK25 (YSK1) | STE20 | STE | 2xik | A | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | |
| STK25 (YSK1) | STE20 | STE | 4nzw | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | | |
| STK25 (YSK1) | STE20 | STE | 7z4v | A | A | ~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamide | Human | Show | |
| STK25 (YSK1) | STE20 | STE | 7z4v | A | B | ~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamide | Human | Show | |
| STK26 (MST4) | STE20 | STE | 3ggf | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | Show | |
