Browse kinase entries (page 261 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
Stk39 (STLK3)STE20STE5dbxBBphosphoaminophosphonic acid-adenylate esterMouseShow
STK4 (MST1)STE20STE3comA-HumanShow
STK4 (MST1)STE20STE3comB-HumanShow
STK4 (MST1)STE20STE6yatA4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHumanShow
STK4 (MST1)STE20STE6yatB4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHumanShow
STK4 (MST1)STE20STE8a5jAA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHumanShow
STK4 (MST1)STE20STE8a5jAB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHumanShow
STK4 (MST1)STE20STE8pavAA1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)ureaHumanShow
STK4 (MST1)STE20STE8pavAB1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)ureaHumanShow
STK4 (MST1)STE20STE8pawA1-[3,5-bis(fluoranyl)-4-[[3-(1-propan-2-ylpyrazol-3-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)ureaHumanShow
STK40 (SgK495)SgK495CAMK5l2qAA-HumanShow
STK40 (SgK495)SgK495CAMK5l2qAB-HumanShow
STK40 (SgK495)SgK495CAMK5l2qBA-HumanShow
STK40 (SgK495)SgK495CAMK5l2qBB-HumanShow
STK40 (SgK495)SgK495CAMK5l2qCA-HumanShow
STK40 (SgK495)SgK495CAMK5l2qCB-HumanShow
STK40 (SgK495)SgK495CAMK5l2qDA-HumanShow
STK40 (SgK495)SgK495CAMK5l2qDB-HumanShow
STRADA (STLK5)STE20STE2wtkBphosphoaminophosphonic acid-adenylate esterHumanShow
STRADA (STLK5)STE20STE2wtkEphosphoaminophosphonic acid-adenylate esterHumanShow
STRADA (STLK5)STE20STE3gniBadenosine-5'-triphosphateHumanShow
STRADA (STLK5)STE20STE8vsuC-HumanShow
SYKSykTK1xbaA-HumanShow
SYKSykTK1xbbAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHumanShow
SYKSykTK1xbbAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHumanShow
SYKSykTK1xbcAAstaurosporineHumanShow
SYKSykTK1xbcABstaurosporineHumanShow
SYKSykTK3emgA2-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-methylethyl]-4-methyl-1,3-thiazole-5-carboxamideHumanShow
SYKSykTK3fqeA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]pyrimidine-5-carboxamideHumanShow
SYKSykTK3fqhAn-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamideHumanShow
SYKSykTK3fqhBn-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamideHumanShow
SYKSykTK3fqsAA6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHumanShow
SYKSykTK3fqsAB6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHumanShow
SYKSykTK3srvAA2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHumanShow
SYKSykTK3srvAB2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHumanShow
SYKSykTK3srvBA2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHumanShow
SYKSykTK3srvBB2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHumanShow
SYKSykTK3tubA1-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-3-[(1r,2s)-2-phenylcyclopropyl]ureaHumanShow
SYKSykTK3tucA1-benzyl-n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-2-oxo-1,2-dihydropyridine-3-carboxamideHumanShow
SYKSykTK3tudAn-{4-methyl-3-[8-methyl-7-oxo-2-(phenylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]phenyl}-3-(trifluoromethyl)benzamideHumanShow
SYKSykTK3vf8A3-[5-(5-ethoxy-6-fluoro-1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]-1,1-diethylureaHumanShow
SYKSykTK3vf9A3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHumanShow
SYKSykTK4dflA3-amino-6-{3-[(methylsulfonyl)amino]phenyl}-n-(piperidin-4-ylmethyl)pyrazine-2-carboxamideHumanShow
SYKSykTK4dfnAA3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamideHumanShow
SYKSykTK4dfnAB3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamideHumanShow
SYKSykTK4f4pAAn-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amineHumanShow
SYKSykTK4f4pABn-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amineHumanShow
SYKSykTK4fl1AAphosphoaminophosphonic acid-adenylate esterHumanShow
SYKSykTK4fl1ABphosphoaminophosphonic acid-adenylate esterHumanShow
SYKSykTK4fl2Aphosphoaminophosphonic acid-adenylate esterHumanShow
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