PDB-code
Browse kinase entries (page 261 of 282)
First 257 258 259 PreviousLast265 264 263 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | Stk39 (STLK3) | STE20 | STE | 5dbx | B | B | phosphoaminophosphonic acid-adenylate ester | Mouse | Show | ![]() |
![]() | STK4 (MST1) | STE20 | STE | 3com | A | - | Human | Show | ![]() | |
![]() | STK4 (MST1) | STE20 | STE | 3com | B | - | Human | Show | ![]() | |
![]() | STK4 (MST1) | STE20 | STE | 6yat | A | 4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine | Human | Show | ![]() | |
![]() | STK4 (MST1) | STE20 | STE | 6yat | B | 4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine | Human | Show | ![]() | |
![]() | STK4 (MST1) | STE20 | STE | 8a5j | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | STK4 (MST1) | STE20 | STE | 8a5j | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | STK4 (MST1) | STE20 | STE | 8pav | A | A | 1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | Show | ![]() |
![]() | STK4 (MST1) | STE20 | STE | 8pav | A | B | 1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | Show | ![]() |
![]() | STK4 (MST1) | STE20 | STE | 8paw | A | 1-[3,5-bis(fluoranyl)-4-[[3-(1-propan-2-ylpyrazol-3-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | Show | ![]() | |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | A | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | B | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | A | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | B | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | A | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | B | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | A | - | Human | Show | ![]() |
![]() | STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | B | - | Human | Show | ![]() |
![]() | STRADA (STLK5) | STE20 | STE | 2wtk | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | STRADA (STLK5) | STE20 | STE | 2wtk | E | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | STRADA (STLK5) | STE20 | STE | 3gni | B | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | STRADA (STLK5) | STE20 | STE | 8vsu | C | - | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 1xba | A | - | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 1xbb | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 1xbb | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 1xbc | A | A | staurosporine | Human | Show | ![]() |
![]() | SYK | Syk | TK | 1xbc | A | B | staurosporine | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3emg | A | 2-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-methylethyl]-4-methyl-1,3-thiazole-5-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3fqe | A | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]pyrimidine-5-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3fqh | A | n-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3fqh | B | n-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3fqs | A | A | 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-one | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3fqs | A | B | 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-one | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3srv | A | A | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3srv | A | B | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3srv | B | A | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3srv | B | B | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 3tub | A | 1-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-3-[(1r,2s)-2-phenylcyclopropyl]urea | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3tuc | A | 1-benzyl-n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3tud | A | n-{4-methyl-3-[8-methyl-7-oxo-2-(phenylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]phenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3vf8 | A | 3-[5-(5-ethoxy-6-fluoro-1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]-1,1-diethylurea | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 3vf9 | A | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 4dfl | A | 3-amino-6-{3-[(methylsulfonyl)amino]phenyl}-n-(piperidin-4-ylmethyl)pyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | SYK | Syk | TK | 4dfn | A | A | 3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4dfn | A | B | 3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4f4p | A | A | n-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amine | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4f4p | A | B | n-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amine | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4fl1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4fl1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | SYK | Syk | TK | 4fl2 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |


