PDB-code
Browse kinase entries (page 52 of 282)
First 48 49 50 PreviousLast56 55 54 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK2 | CDK | CMGC | 5anj | A | n-(9h-purin-6-yl)thiophene-2-carboxamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5ank | A | 2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5ano | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5cyi | A | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5cyi | A | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5cyi | C | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5cyi | C | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5d1j | A | n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5fp5 | A | 4-fluorobenzoic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5fp6 | A | A | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5fp6 | A | B | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iev | A | A | roniciclib | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iev | A | B | roniciclib | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iex | A | A | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iex | A | B | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iey | A | A | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5iey | A | B | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5if1 | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5if1 | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5if1 | C | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5if1 | C | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5jq5 | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5jq8 | A | (3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5k4j | A | A | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5k4j | A | B | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5l2w | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5lmk | A | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5lmk | A | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5lmk | C | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5lmk | C | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5mhq | A | A | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5mhq | A | B | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5nev | A | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5nev | C | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5oo0 | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5oo0 | A | C | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5oo1 | A | ~{n}-(4-pyrimidin-2-ylphenyl)propanamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5oo3 | A | A | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5oo3 | A | B | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5osj | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5osj | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5osm | A | A | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5osm | A | B | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 5uq1 | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5uq1 | C | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5uq2 | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 5uq3 | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 6ath | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6ath | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6gub | A | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | Show | ![]() |


