Browse kinase entries (page 52 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC5anjAn-(9h-purin-6-yl)thiophene-2-carboxamideHumanShow
CDK2CDKCMGC5ankA2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamideHumanShow
CDK2CDKCMGC5anoA-HumanShow
CDK2CDKCMGC5cyiAA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHumanShow
CDK2CDKCMGC5cyiAB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHumanShow
CDK2CDKCMGC5cyiCA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHumanShow
CDK2CDKCMGC5cyiCB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHumanShow
CDK2CDKCMGC5d1jAn-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamideHumanShow
CDK2CDKCMGC5fp5A4-fluorobenzoic acidHumanShow
CDK2CDKCMGC5fp6AA3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHumanShow
CDK2CDKCMGC5fp6AB3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHumanShow
CDK2CDKCMGC5ievAAroniciclibHumanShow
CDK2CDKCMGC5ievABroniciclibHumanShow
CDK2CDKCMGC5iexAA(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHumanShow
CDK2CDKCMGC5iexAB(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHumanShow
CDK2CDKCMGC5ieyAA4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHumanShow
CDK2CDKCMGC5ieyAB4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHumanShow
CDK2CDKCMGC5if1AA-HumanShow
CDK2CDKCMGC5if1AB-HumanShow
CDK2CDKCMGC5if1CA-HumanShow
CDK2CDKCMGC5if1CB-HumanShow
CDK2CDKCMGC5jq5A(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK2CDKCMGC5jq8A(3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK2CDKCMGC5k4jAA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHumanShow
CDK2CDKCMGC5k4jAB1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHumanShow
CDK2CDKCMGC5l2wA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHumanShow
CDK2CDKCMGC5lmkAA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHumanShow
CDK2CDKCMGC5lmkAB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHumanShow
CDK2CDKCMGC5lmkCA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHumanShow
CDK2CDKCMGC5lmkCB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHumanShow
CDK2CDKCMGC5mhqAA(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHumanShow
CDK2CDKCMGC5mhqAB(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHumanShow
CDK2CDKCMGC5nevA4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC5nevC4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC5oo0AA-HumanShow
CDK2CDKCMGC5oo0AC-HumanShow
CDK2CDKCMGC5oo1A~{n}-(4-pyrimidin-2-ylphenyl)propanamideHumanShow
CDK2CDKCMGC5oo3AA1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHumanShow
CDK2CDKCMGC5oo3AB1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHumanShow
CDK2CDKCMGC5osjAA-HumanShow
CDK2CDKCMGC5osjAB-HumanShow
CDK2CDKCMGC5osmAAmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHumanShow
CDK2CDKCMGC5osmABmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHumanShow
CDK2CDKCMGC5uq1A-HumanShow
CDK2CDKCMGC5uq1C-HumanShow
CDK2CDKCMGC5uq2A-HumanShow
CDK2CDKCMGC5uq3A-HumanShow
CDK2CDKCMGC6athAA-HumanShow
CDK2CDKCMGC6athAB-HumanShow
CDK2CDKCMGC6gubA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHumanShow
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