Browse kinase entries (page 54 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC6q4fACpyridine-2,6-diamineHumanShow
CDK2CDKCMGC6q4gAA2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4gAB2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4hAA2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4hAB2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4iAA2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4iAB2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4jAA2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4jAB2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHumanShow
CDK2CDKCMGC6q4kAA-HumanShow
CDK2CDKCMGC6q4kAB-HumanShow
CDK2CDKCMGC6q4kAC-HumanShow
CDK2CDKCMGC6rijAA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHumanShow
CDK2CDKCMGC6rijAB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHumanShow
CDK2CDKCMGC6rijCA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHumanShow
CDK2CDKCMGC6rijCB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHumanShow
CDK2CDKCMGC6sg4AA-HumanShow
CDK2CDKCMGC6sg4AB-HumanShow
CDK2CDKCMGC6sg4CA-HumanShow
CDK2CDKCMGC6sg4CB-HumanShow
CDK2CDKCMGC6yl1AAmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHumanShow
CDK2CDKCMGC6yl1ABmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHumanShow
CDK2CDKCMGC6yl6AA-HumanShow
CDK2CDKCMGC6yl6AB-HumanShow
CDK2CDKCMGC6ylkAAmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHumanShow
CDK2CDKCMGC6ylkABmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHumanShow
CDK2CDKCMGC7ackAA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHumanShow
CDK2CDKCMGC7ackAB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHumanShow
CDK2CDKCMGC7ackCA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHumanShow
CDK2CDKCMGC7ackCB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHumanShow
CDK2CDKCMGC7b5lL-HumanShow
CDK2CDKCMGC7b5rL-HumanShow
CDK2CDKCMGC7b7sAA7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHumanShow
CDK2CDKCMGC7b7sAB7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHumanShow
CDK2CDKCMGC7e34A-HumanShow
CDK2CDKCMGC7kjsA6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
CDK2CDKCMGC7m2fAA[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHumanShow
CDK2CDKCMGC7m2fAB[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHumanShow
CDK2CDKCMGC7mkxA2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamideHumanShow
CDK2CDKCMGC7nvqAstaurosporineHumanShow
CDK2CDKCMGC7qhlAA5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHumanShow
CDK2CDKCMGC7qhlAB5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHumanShow
CDK2CDKCMGC7ra5AA4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC7ra5AB4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC7rweA5-nitro-2-[(3-phenylpropyl)amino]benzoic acidHumanShow
CDK2CDKCMGC7rwfA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHumanShow
CDK2CDKCMGC7rxoAA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHumanShow
CDK2CDKCMGC7rxoAB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHumanShow
CDK2CDKCMGC7s4tAA2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHumanShow
CDK2CDKCMGC7s4tAB2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHumanShow
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