PDB-code
Browse kinase entries (page 54 of 282)
First 50 51 52 PreviousLast58 57 56 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK2 | CDK | CMGC | 6q4f | A | C | pyridine-2,6-diamine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4g | A | A | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4g | A | B | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4h | A | A | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4h | A | B | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4i | A | A | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4i | A | B | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4j | A | A | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4j | A | B | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4k | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4k | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6q4k | A | C | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6rij | A | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6rij | A | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6rij | C | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6rij | C | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6sg4 | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6sg4 | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6sg4 | C | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6sg4 | C | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6yl1 | A | A | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6yl1 | A | B | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6yl6 | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6yl6 | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6ylk | A | A | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 6ylk | A | B | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ack | A | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ack | A | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ack | C | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ack | C | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7b5l | L | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7b5r | L | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7b7s | A | A | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7b7s | A | B | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7e34 | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7kjs | A | 6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7m2f | A | A | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7m2f | A | B | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7mkx | A | 2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7nvq | A | staurosporine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7qhl | A | A | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7qhl | A | B | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ra5 | A | A | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ra5 | A | B | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7rwe | A | 5-nitro-2-[(3-phenylpropyl)amino]benzoic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7rwf | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7rxo | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7rxo | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s4t | A | A | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s4t | A | B | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | Show | ![]() |


