PDB-code
Browse kinase entries (page 60 of 282)
First 56 57 58 PreviousLast64 63 62 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | CHEK1 (CHK1) | CAMKL | CAMK | 2qhn | A | 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one | Human | Show |  | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2r0u | A | 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmq | A | n-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | A | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | B | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wms | A | [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | A | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | B | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | A | 6-morpholin-4-yl-9h-purine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | B | 6-morpholin-4-yl-9h-purine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmv | A | 1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmw | A | 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmx | A | 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | A | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | B | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8e | A | 5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | A | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | B | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xey | A | 3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xez | A | 6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xf0 | A | 3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | A | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | B | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | A | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | B | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydk | A | 2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | A | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | B | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | A | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | B | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | A | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | B | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | A | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | B | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym5 | A | (3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | A | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | B | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | A | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | B | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym8 | A | (r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ywp | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | A | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | B | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvr | A | - | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvs | A | - | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3nlb | A | 3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | A | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | B | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | A | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | B | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
