PDB-code
Browse kinase entries (page 10 of 282)
First 6 7 8 PreviousLast14 13 12 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | ACVR2A (ACTR2) | STKR | TKL | 4asx | A | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | Show |  |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | A | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | Show | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | Show | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | Show | |
| ACVR2B (ACTR2B) | STKR | TKL | 2qlu | A | adenine | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | C | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | D | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | E | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | F | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | G | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | H | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | I | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | J | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | K | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | L | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | M | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | N | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | O | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | P | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | Q | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | R | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | S | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | T | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | U | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | V | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | W | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | X | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | | |
| AKT1 | Akt | AGC | 3cqu | A | A | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| AKT1 | Akt | AGC | 3cqu | A | B | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| AKT1 | Akt | AGC | 3cqw | A | A | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | Show | |
| AKT1 | Akt | AGC | 3cqw | A | B | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | Show | |
| AKT1 | Akt | AGC | 3mv5 | A | A | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | Show | |
| AKT1 | Akt | AGC | 3mv5 | A | B | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | Show | |
| AKT1 | Akt | AGC | 3mvh | A | A | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | Show | |
| AKT1 | Akt | AGC | 3mvh | A | B | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | Show | |
| AKT1 | Akt | AGC | 3o96 | A | - | Human | Show | | |
| AKT1 | Akt | AGC | 3ocb | A | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | Show | | |
| AKT1 | Akt | AGC | 3ocb | B | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | Show | | |
| AKT1 | Akt | AGC | 3ow4 | A | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | Show | | |
| AKT1 | Akt | AGC | 3ow4 | B | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | Show | | |
| AKT1 | Akt | AGC | 3qkk | A | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | Show | | |
| AKT1 | Akt | AGC | 3qkl | A | n-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamide | Human | Show | | |
| AKT1 | Akt | AGC | 3qkm | A | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | Show | | |
| AKT1 | Akt | AGC | 4ejn | A | - | Human | Show | | |
| AKT1 | Akt | AGC | 4ekk | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| AKT1 | Akt | AGC | 4ekk | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| AKT1 | Akt | AGC | 4ekl | A | (2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-one | Human | Show | | |
| AKT1 | Akt | AGC | 4gv1 | A | A | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | Show | |
