PDB-code
Browse kinase entries (page 91 of 282)
First 87 88 89 PreviousLast95 94 93 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | DCLK1 | DCAMKL | CAMK | 5jzj | A | B | amp phosphoramidate | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 5jzj | B | A | amp phosphoramidate | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 5jzj | B | B | amp phosphoramidate | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 5jzn | A | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 5jzn | B | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 6kyq | A | A | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyq | A | B | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyq | B | A | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyq | B | B | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyr | A | A | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyr | A | B | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyr | B | A | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 6kyr | B | B | - | Human | Show | ![]() |
![]() | DCLK1 | DCAMKL | CAMK | 7f3g | A | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 7kx6 | A | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 7kx8 | A | 5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 7kxw | A | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | DCLK1 | DCAMKL | CAMK | 7kxw | B | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 3zos | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 3zos | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 3zos | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 3zos | B | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4bkj | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4bkj | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4bkj | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4bkj | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4ckr | A | A | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 4ckr | A | B | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5bvk | A | 1-(2-chlorophenyl)-3-(pyridin-3-ylmethyl)urea | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5bvn | A | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5bvo | A | n-(5-{(1s)-1-[(5-fluoro-1,3-benzoxazol-2-yl)amino]ethyl}-2-methylphenyl)imidazo[1,2-a]pyridine-3-carboxamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5bvw | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5fdp | A | (4~{s})-4-methyl-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinoline-7-carboxamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5fdx | A | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5fdx | B | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5sau | A | A | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sau | A | B | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sav | A | A | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sav | A | B | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5saw | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5saw | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sax | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sax | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5say | A | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5saz | A | A | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5saz | A | B | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sb0 | A | n-{[(1r,2s)-2-{2-[(pyridin-3-yl)oxy]ethyl}cyclohexyl]methyl}-3-(trifluoromethoxy)benzamide | Human | Show | ![]() | |
![]() | DDR1 | DDR | TK | 5sb1 | A | A | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sb1 | A | B | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | Show | ![]() |
![]() | DDR1 | DDR | TK | 5sb2 | A | A | 3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | Show | ![]() |


