PDB-code
Search results (20 entries covering 7 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | FGFR4 | FGFR | TK | 4tyi | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 5a46 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | STK10 (LOK) | STE20 | STE | 5owq | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am7 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am7 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am6 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am6 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am7 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5a46 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am6 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5a46 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am6 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5am7 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 5a46 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | EIF2AK4 (GCN2) | PEK | Other | 7qq6 | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() | |
![]() | STK17B (DRAK2) | DAPK | CAMK | 7akg | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | STK17B (DRAK2) | DAPK | CAMK | 7akg | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | STK10 (LOK) | STE20 | STE | 5owq | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | STK10 (LOK) | STE20 | STE | 5owq | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |
![]() | STK10 (LOK) | STE20 | STE | 5owq | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | Show | ![]() |


