Search results (16 entries covering 7 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DAPK3DAPKCAMK2j90AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
DAPK3DAPKCAMK2j90BA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
Jak2 (JAK2)JakATK4gl9D2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouseShow
Jak2 (JAK2)JakATK4gl9B2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouseShow
Jak2 (JAK2)JakATK4gl9C2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouseShow
Jak2 (JAK2)JakATK4gl9A2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouseShow
JAK1JakATK3eyhA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
JAK3JakATK3lxlAB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
JAK3JakATK3lxlAA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
JAK2JakATK2b7aB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
JAK2JakATK2b7aA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
TYK2JakATK3lxpA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
TYK2JakATK3nz0AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
DAPK3DAPKCAMK2j90BB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
DAPK3DAPKCAMK2j90AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow
TYK2JakATK3nz0AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHumanShow