PDB-code
Search results (16 entries covering 7 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | DAPK3 | DAPK | CAMK | 2j90 | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | DAPK3 | DAPK | CAMK | 2j90 | B | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | Jak2 (JAK2) | JakA | TK | 4gl9 | D | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | Show | ![]() | |
![]() | Jak2 (JAK2) | JakA | TK | 4gl9 | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | Show | ![]() | |
![]() | Jak2 (JAK2) | JakA | TK | 4gl9 | C | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | Show | ![]() | |
![]() | Jak2 (JAK2) | JakA | TK | 4gl9 | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | Show | ![]() | |
![]() | JAK1 | JakA | TK | 3eyh | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() | |
![]() | JAK3 | JakA | TK | 3lxl | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | JAK3 | JakA | TK | 3lxl | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | JAK2 | JakA | TK | 2b7a | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() | |
![]() | JAK2 | JakA | TK | 2b7a | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() | |
![]() | TYK2 | JakA | TK | 3lxp | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() | |
![]() | TYK2 | JakA | TK | 3nz0 | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | DAPK3 | DAPK | CAMK | 2j90 | B | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | DAPK3 | DAPK | CAMK | 2j90 | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |
![]() | TYK2 | JakA | TK | 3nz0 | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | Show | ![]() |


