Search results (38 entries covering 4 PDB structures)

Your browser unfortunately does not support an HTML5 canvas. Your browser unfortunately does not support an HTML5 canvas.
#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
BMPR1BSTKRTKL3mdyCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
BMPR1BSTKRTKL3mdyCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
BMPR1BSTKRTKL3mdyAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0I4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0N4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0J4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0G4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0C4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0S4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0R4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0T4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0A4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0O4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0L4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0M4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0V4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0E4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0H4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0D4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0B4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0X4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0P4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
BMPR1BSTKRTKL3mdyAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0F4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0Q4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0U4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0W4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVRL1 (ALK1)STKRTKL3my0K4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uBA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL6unsAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL6unsAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uDB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uBB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow
ACVR1 (ALK2)STKRTKL3q4uDA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHumanShow