PDB-code
Search results (38 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | BMPR1B | STKR | TKL | 3mdy | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | BMPR1B | STKR | TKL | 3mdy | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | BMPR1B | STKR | TKL | 3mdy | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | I | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | N | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | J | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | G | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | C | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | S | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | R | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | T | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | O | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | L | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | M | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | V | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | E | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | H | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | D | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | X | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | P | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | BMPR1B | STKR | TKL | 3mdy | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | F | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | Q | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | U | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | W | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVRL1 (ALK1) | STKR | TKL | 3my0 | K | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() | |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | B | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 6uns | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 6uns | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | D | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | B | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 3q4u | D | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | Show | ![]() |


