Search results (11 entries covering 5 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MARK2CAMKLCAMK5kz7A7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHumanShow
MARK2CAMKLCAMK5kz8A5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHumanShow
MARK2CAMKLCAMK5eakAn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHumanShow
MARK2CAMKLCAMK3iecA-HumanShow
MARK2CAMKLCAMK5kz7B7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHumanShow
MARK2CAMKLCAMK5kz8B5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHumanShow
MARK2CAMKLCAMK3iecC-HumanShow
MARK2CAMKLCAMK5eakBn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHumanShow
MARK2CAMKLCAMK3iecB-HumanShow
MARK2CAMKLCAMK3iecD-HumanShow
MARK2CAMKLCAMK8txyAn-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamideHumanShow