Search results (66 entries covering 31 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
HASPIN (Haspin)HaspinOther6z56AC6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
HASPIN (Haspin)HaspinOther6g37AB5-fluorotubercidinHumanShow
HASPIN (Haspin)HaspinOther4qtcAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHumanShow
HASPIN (Haspin)HaspinOther6z5dAB11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one HumanShow
HASPIN (Haspin)HaspinOther6z5bAA6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
HASPIN (Haspin)HaspinOther6g3aAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6g38AB'2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther2vuwAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther2wb8AB-HumanShow
HASPIN (Haspin)HaspinOther7opsA2-methylsulfanyl-10-nitro-pyrido[3,4-g]quinazolineHumanShow
HASPIN (Haspin)HaspinOther7sqmAA1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amineHumanShow
HASPIN (Haspin)HaspinOther6g34AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6g39AC-HumanShow
HASPIN (Haspin)HaspinOther6z56AB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
HASPIN (Haspin)HaspinOther6z5bAB6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
HASPIN (Haspin)HaspinOther8rdkA3-pyridin-4-yl-1~{h}-pyrrolo[3,2-g]isoquinolineHumanShow
HASPIN (Haspin)HaspinOther6g38AA'2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6g35AA5-bromotubercidinHumanShow
HASPIN (Haspin)HaspinOther6z5aABn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide HumanShow
HASPIN (Haspin)HaspinOther6g35AD-HumanShow
HASPIN (Haspin)HaspinOther3fmdABn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHumanShow
HASPIN (Haspin)HaspinOther6z59AB11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHumanShow
HASPIN (Haspin)HaspinOther4oucAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther3f2nAB(2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-olHumanShow
HASPIN (Haspin)HaspinOther6z5eAA11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one HumanShow
HASPIN (Haspin)HaspinOther6z5cAB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
HASPIN (Haspin)HaspinOther7sqmAB1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amineHumanShow
HASPIN (Haspin)HaspinOther6g39AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6z5cAA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
HASPIN (Haspin)HaspinOther5htbAA-HumanShow
HASPIN (Haspin)HaspinOther6z57AA10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaeneHumanShow
HASPIN (Haspin)HaspinOther3f2nAA(2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-olHumanShow
HASPIN (Haspin)HaspinOther6g37AA5-fluorotubercidinHumanShow
HASPIN (Haspin)HaspinOther6z56AA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
HASPIN (Haspin)HaspinOther7avqAB(2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olHumanShow
HASPIN (Haspin)HaspinOther6z57AB10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaeneHumanShow
HASPIN (Haspin)HaspinOther2vuwAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther5htcAB-HumanShow
HASPIN (Haspin)HaspinOther3e7vAA3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amineHumanShow
HASPIN (Haspin)HaspinOther6g36AB5-chlorotubercidinHumanShow
HASPIN (Haspin)HaspinOther3dlzABadenosine monophosphateHumanShow
HASPIN (Haspin)HaspinOther5htcAC-HumanShow
HASPIN (Haspin)HaspinOther6g36AA5-chlorotubercidinHumanShow
HASPIN (Haspin)HaspinOther6g35AB5-bromotubercidinHumanShow
HASPIN (Haspin)HaspinOther6g3aAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther5htbAB-HumanShow
HASPIN (Haspin)HaspinOther5htcAA-HumanShow
HASPIN (Haspin)HaspinOther6g39AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6z5dAA11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one HumanShow
HASPIN (Haspin)HaspinOther6z59AA11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHumanShow
HASPIN (Haspin)HaspinOther2wb8AA-HumanShow
HASPIN (Haspin)HaspinOther3e7vAB3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amineHumanShow
HASPIN (Haspin)HaspinOther6z58AA8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHumanShow
HASPIN (Haspin)HaspinOther6g39AD-HumanShow
HASPIN (Haspin)HaspinOther3iq7AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther6g35AC-HumanShow
HASPIN (Haspin)HaspinOther6z5aAAn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide HumanShow
HASPIN (Haspin)HaspinOther4oucAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther7avqAA(2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olHumanShow
HASPIN (Haspin)HaspinOther6z5eAB11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one HumanShow
HASPIN (Haspin)HaspinOther3fmdAAn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHumanShow
HASPIN (Haspin)HaspinOther6g34AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther3dlzAAadenosine monophosphateHumanShow
HASPIN (Haspin)HaspinOther6z58AB8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHumanShow
HASPIN (Haspin)HaspinOther4qtcAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHumanShow
HASPIN (Haspin)HaspinOther3iq7AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow