PDB-code
Browse kinase entries (page 120 of 282)
First 116 117 118 PreviousLast124 123 122 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | FGFR1 | FGFR | TK | 3kxx | B | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3kxx | C | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3kxx | D | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3ky2 | A | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3ky2 | B | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3rhx | A | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3rhx | B | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3tt0 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3tt0 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3tt0 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3tt0 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f63 | A | 5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4f63 | B | 5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4f64 | A | A | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f64 | A | B | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f64 | B | A | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f64 | B | B | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f65 | A | A | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f65 | A | B | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f65 | B | A | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4f65 | B | B | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4nk9 | A | n~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4nk9 | B | n~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4nka | A | n~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4nka | B | n~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4nks | A | A | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4nks | A | B | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4nks | B | A | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4nks | B | B | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwi | A | A | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwi | A | B | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwi | B | A | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwi | B | B | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwj | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwj | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwj | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwj | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwk | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwk | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwk | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwk | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4rwl | A | - | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4rwl | B | 6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamide | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 4uwb | A | A | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwb | A | B | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwb | B | A | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwb | B | B | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwc | A | A | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwc | A | B | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 4uwc | B | A | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | Show | ![]() |


