Browse kinase entries (page 120 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
FGFR1FGFRTK3kxxB-HumanShow
FGFR1FGFRTK3kxxC-HumanShow
FGFR1FGFRTK3kxxD-HumanShow
FGFR1FGFRTK3ky2A-HumanShow
FGFR1FGFRTK3ky2B-HumanShow
FGFR1FGFRTK3rhxA(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHumanShow
FGFR1FGFRTK3rhxB(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHumanShow
FGFR1FGFRTK3tt0AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK3tt0AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK3tt0BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK3tt0BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK4f63A5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f63B5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f64AA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f64AB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f64BA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f64BB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f65AA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f65AB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f65BA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4f65BB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nk9An~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nk9Bn~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nkaAn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nkaBn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nksAAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nksABn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nksBAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nksBBn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4rwiAA-HumanShow
FGFR1FGFRTK4rwiAB-HumanShow
FGFR1FGFRTK4rwiBA-HumanShow
FGFR1FGFRTK4rwiBB-HumanShow
FGFR1FGFRTK4rwjAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwjABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwjBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwjBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwkAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwkABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwkBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwkBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4rwlA-HumanShow
FGFR1FGFRTK4rwlB6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamideHumanShow
FGFR1FGFRTK4uwbAAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK4uwbABn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK4uwbBAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK4uwbBBn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK4uwcAA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK4uwcAB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK4uwcBA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
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