PDB-code
Browse kinase entries (page 175 of 282)
First 171 172 173 PreviousLast179 178 177 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4h3p | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4h3p | D | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4h3q | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | B | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | C | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | D | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | A | caffeic acid | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | B | caffeic acid | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | A | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | B | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | A | n-benzyl-9h-purin-6-amine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | B | n-benzyl-9h-purin-6-amine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | A | 5-chloro-1,3-benzoxazol-2-amine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | B | - | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | A | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | B | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | A | n-cyclohexyl-9h-purin-6-amine | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | B | n-cyclohexyl-9h-purin-6-amine | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | A | n-cyclohexyl-9h-purin-6-amine | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | B | n-cyclohexyl-9h-purin-6-amine | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | A | 5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | B | 5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | A | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | B | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | A | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | B | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qp9 | A | 7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qpa | A | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qpa | B | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | A | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | B | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | A | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | B | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | A | catechol | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | B | catechol | Human | Show | ![]() |


