PDB-code
Browse kinase entries (page 208 of 282)
First 204 205 206 PreviousLast212 211 210 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MTOR (FRAP) | PIKK | Atypical | 9f44 | A | - | Human | Show | ![]() | |
![]() | MTOR (FRAP) | PIKK | Atypical | 9f45 | A | - | Human | Show | ![]() | |
![]() | MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4apc | A | A | - | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4apc | A | B | - | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4apc | B | A | - | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4apc | B | B | - | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4b9d | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4b9d | A | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4b9d | B | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | Show | ![]() |
![]() | NEK1 | NEK | Other | 4b9d | B | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2jav | A | A | 5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2jav | A | B | 5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5a | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5a | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5b | A | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5b | A | B | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5h | A | A | - | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2w5h | A | B | - | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2wqo | A | 4-[2-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]benzoic acid | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 2xk3 | A | A | 4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk3 | A | B | 4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk4 | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk4 | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk4 | A | C | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk6 | A | cis-4-[3-amino-6-(3-cyclopropylthiophen-2-yl)pyrazin-2-yl]cyclohexanecarboxylic acid | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 2xk7 | A | A | (3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk7 | A | B | (3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xk8 | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methoxybenzoic acid | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 2xkc | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xkc | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xkd | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xkd | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xke | A | 1-[3-amino-6-(3-methoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 2xkf | A | A | 1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xkf | A | B | 1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnm | A | A | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnm | A | B | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnn | A | A | 5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnn | A | B | 5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xno | A | A | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xno | A | B | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnp | A | A | 4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 2xnp | A | B | 4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | Show | ![]() |
![]() | NEK2 | NEK | Other | 4a4x | A | 4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 4afe | A | 4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{[(1r,2z)-4,4,4-trifluoro-1-methylbut-2-en-1-yl]oxy}benzamide | Human | Show | ![]() | |
![]() | NEK2 | NEK | Other | 5m51 | A | 3-[[6-(cyclohexylmethoxy)-9~{h}-purin-2-yl]amino]benzamide | Human | Show | ![]() |


