Browse kinase entries (page 252 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
ROCK2DMPKAGC7jntCBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntDAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntDBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntEAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntEBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntFAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntFBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntGAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntGBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntHAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jntHBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHumanShow
ROCK2DMPKAGC7jovAn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovBn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovCn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovDn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovEn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovFn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovGn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7jovHn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHumanShow
ROCK2DMPKAGC7p6nA~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-piperidine-1-carboxamideHumanShow
ROCK2DMPKAGC8gdsA4-{4-[2-(2,3-dihydro-1h-indol-1-yl)-2-oxoethyl]phenyl}phthalazin-1(2h)-oneHumanShow
ROR1RorTK6tu9A3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
ROR1RorTK6tu9B3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
ROR2RorTK3zzwAA-HumanShow
ROR2RorTK3zzwAB-HumanShow
ROR2RorTK3zzwBA-HumanShow
ROR2RorTK3zzwBB-HumanShow
ROR2RorTK4gt4AA-HumanShow
ROR2RorTK4gt4AB-HumanShow
ROR2RorTK4gt4BA-HumanShow
ROR2RorTK4gt4BB-HumanShow
ROS1 (ROS)SevTK3zbfA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHumanShow
ROS1 (ROS)SevTK4uxlA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHumanShow
ROS1 (ROS)SevTK7z5wA~{n}-[6-methyl-2-[(2~{s})-2-[3-(3-methylpyrazin-2-yl)-1,2-oxazol-5-yl]pyrrolidin-1-yl]pyrimidin-4-yl]-1,3-thiazol-2-amineHumanShow
ROS1 (ROS)SevTK7z5xA(2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diolHumanShow
RPS6KA1 (RSK3)RSKAGC2z7qAphosphomethylphosphonic acid adenylate esterHumanShow
RPS6KA1 (RSK3)RSKAGC2z7rAstaurosporineHumanShow
RPS6KA1 (RSK3)RSKAGC2z7sA2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAB-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBB-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAB-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBB-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAB-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDA-HumanShow
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDB-HumanShow
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