PDB-code
Browse kinase entries (page 252 of 282)
First 248 249 250 PreviousLast256 255 254 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | ROCK2 | DMPK | AGC | 7jnt | C | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | D | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | D | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | E | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | E | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | F | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | F | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | G | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | G | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | H | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jnt | H | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | Show | ![]() |
![]() | ROCK2 | DMPK | AGC | 7jov | A | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | B | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | C | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | D | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | E | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | F | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | G | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7jov | H | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 7p6n | A | ~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-piperidine-1-carboxamide | Human | Show | ![]() | |
![]() | ROCK2 | DMPK | AGC | 8gds | A | 4-{4-[2-(2,3-dihydro-1h-indol-1-yl)-2-oxoethyl]phenyl}phthalazin-1(2h)-one | Human | Show | ![]() | |
![]() | ROR1 | Ror | TK | 6tu9 | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() | |
![]() | ROR1 | Ror | TK | 6tu9 | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | Show | ![]() | |
![]() | ROR2 | Ror | TK | 3zzw | A | A | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 3zzw | A | B | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 3zzw | B | A | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 3zzw | B | B | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 4gt4 | A | A | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 4gt4 | A | B | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 4gt4 | B | A | - | Human | Show | ![]() |
![]() | ROR2 | Ror | TK | 4gt4 | B | B | - | Human | Show | ![]() |
![]() | ROS1 (ROS) | Sev | TK | 3zbf | A | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | Show | ![]() | |
![]() | ROS1 (ROS) | Sev | TK | 4uxl | A | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | Show | ![]() | |
![]() | ROS1 (ROS) | Sev | TK | 7z5w | A | ~{n}-[6-methyl-2-[(2~{s})-2-[3-(3-methylpyrazin-2-yl)-1,2-oxazol-5-yl]pyrrolidin-1-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine | Human | Show | ![]() | |
![]() | ROS1 (ROS) | Sev | TK | 7z5x | A | (2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol | Human | Show | ![]() | |
![]() | RPS6KA1 (RSK3) | RSK | AGC | 2z7q | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | RPS6KA1 (RSK3) | RSK | AGC | 2z7r | A | staurosporine | Human | Show | ![]() | |
![]() | RPS6KA1 (RSK3) | RSK | AGC | 2z7s | A | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | Show | ![]() | |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | B | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | B | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | B | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | B | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | B | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | A | - | Human | Show | ![]() |
![]() | RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | B | - | Human | Show | ![]() |


