PDB-code
Search results (27 entries covering 18 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | AKT2 | Akt | AGC | 9c1w | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e88 | B | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e87 | A | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 2jdr | A | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e87 | B | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 3e87 | B | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 1o6k | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 2x39 | A | 4-amino-n-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 1mry | A | - | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 8q61 | A | A | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 8q61 | A | B | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 3e8d | A | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 1gzo | A | - | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e8d | A | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 3d0e | A | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e8d | B | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 3d0e | B | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e8d | B | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 3e87 | A | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | AKT2 | Akt | AGC | 1gzn | A | - | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 1o6l | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 2xh5 | A | 4-(4-tert-butylbenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminium | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 3e88 | A | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 2jdo | A | isoquinoline-5-sulfonic acid (2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)amide | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 1mrv | A | - | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 1gzk | A | - | Human | Show | ![]() | |
![]() | AKT2 | Akt | AGC | 2uw9 | A | 4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidine | Human | Show | ![]() |


