Search results (257 entries covering 80 PDB structures)

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#	Kinase	Family	Group	PDB	Chain	(Alternate) Model	Orthosteric ligand	Organism	Details	File
	DYRK1A	DYRK	CMGC	6eis	C	B	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	C	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6eiv	B		~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	7a52	A	B	3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	A	B	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	C	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	B	A	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	5a4q	A		n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	C	A	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6s17	A	A	~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj4	A	A	4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6uip	A		4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	2wo6	A	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	D	A	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	B	B	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eip	C		4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	A	B	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	6eij	B		~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide	Human	Show
	DYRK1A	DYRK	CMGC	7ak2	A		4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	7a51	A		4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrile	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	B	B	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6ln1	A		1,3,5,8-tetrakis(oxidanyl)xanthen-9-one	Human	Show
	DYRK1A	DYRK	CMGC	6yf8	B		~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	8c3r	A	B	gossypin	Human	Show
	DYRK1A	DYRK	CMGC	8c3r	A	A	gossypin	Human	Show
	DYRK1A	DYRK	CMGC	8c3g	A	A	n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	8c3q	A	B	rutin	Human	Show
	DYRK1A	DYRK	CMGC	8c3g	A	B	n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	8c3q	A	A	rutin	Human	Show
	DYRK1A	DYRK	CMGC	7fhs	A	B	(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	C	A	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	4aze	B		5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one	Human	Show
	DYRK1A	DYRK	CMGC	2wo6	A	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6s11	A	A	6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	3anr	B		7-methoxy-1-methyl-9h-beta-carboline	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	D	B	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6a1f	A	B	8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	6s1j	A	A	3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	6s11	B	B	6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	A	A	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	6eiq	B		[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	6eif	D		4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide	Human	Show
	DYRK1A	DYRK	CMGC	7a53	A	B	(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one	Human	Show
	DYRK1A	DYRK	CMGC	7a5d	A	A	4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile	Human	Show
	DYRK1A	DYRK	CMGC	6ej4	D		3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline	Human	Show
	DYRK1A	DYRK	CMGC	4nct	A		pkc412	Human	Show
	DYRK1A	DYRK	CMGC	5a3x	A		n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7zh8	A	B	6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine	Human	Show
	DYRK1A	DYRK	CMGC	6yf8	D		~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	A	A	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4t	A		n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7aj8	A	A	4-(1-benzofuran-5-yl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7zh8	A	A	6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	D	B	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	C	B	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7a4r	A	B	2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	7akl	A		4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	D	A	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	5aik	D		4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine	Human	Show
	DYRK1A	DYRK	CMGC	7o7k	A	B	n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a3x	C		n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eip	A		4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6eiq	D		[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	7ajm	A	A	~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	A	A	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	7aj5	A	B	4-(1-benzofuran-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	6eip	D		4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	D	A	-	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	B	B	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6a1g	B		5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	B	A	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	C	A	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	4aze	C		5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one	Human	Show
	DYRK1A	DYRK	CMGC	5aik	A		4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj2	A	B	4-(4-methoxyphenyl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6eiv	A		~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	D	A	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	D	A	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	D	B	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	B	B	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1j	A	B	3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	C	B	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	D	A	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	6uip	B		4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6eir	C		~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	7a4o	A		phosphoaminophosphonic acid-adenylate ester	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	C	A	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	C	B	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	A	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	C	A	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	6a1g	A		5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	7a5d	A	B	4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	C	B	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	7ajv	A		4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	7a55	A		3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6eil	A		[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	6eiq	A		[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	6eil	C		-	Human	Show
	DYRK1A	DYRK	CMGC	7a5l	A	A	4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	3anq	D		(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one	Human	Show
	DYRK1A	DYRK	CMGC	7aka	A	B	4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	3anr	A		7-methoxy-1-methyl-9h-beta-carboline	Human	Show
	DYRK1A	DYRK	CMGC	6eis	A	B	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	6eil	B		[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	5a54	A		n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	B	A	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	A	B	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	B	A	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eis	C	A	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	7aka	A	A	4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	4ylk	A	B	10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	3anr	D		7-methoxy-1-methyl-9h-beta-carboline	Human	Show
	DYRK1A	DYRK	CMGC	7aja	A	B	1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine	Human	Show
	DYRK1A	DYRK	CMGC	6s11	B	A	6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	5a4q	C		n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4t	C		n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7ajm	A	B	~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eip	B		4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide	Human	Show
	DYRK1A	DYRK	CMGC	4nct	C		pkc412	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	B	A	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	D	A	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	C	A	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	6ej4	A		3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline	Human	Show
	DYRK1A	DYRK	CMGC	3anr	C		7-methoxy-1-methyl-9h-beta-carboline	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	D	B	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6s17	A	B	~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	C	A	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7a52	A	A	3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	A	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	7ajs	A	A	4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	6eil	D		[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	7a4s	A		7-chlorothieno[3,2-c]pyridin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj7	A		4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	6s1h	A	A	~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6eir	B		~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eis	B	B	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	7ake	A		4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	5a4q	B		n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	D	B	-	Human	Show
	DYRK1A	DYRK	CMGC	6eiv	D		~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eis	D	B	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	6eir	A		~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	A	A	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	A	A	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	7aj5	A	A	4-(1-benzofuran-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	6s1b	A	A	~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj8	A	B	4-(1-benzofuran-5-yl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	C	B	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	5aik	B		4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	C	A	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6eis	B	A	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	7z5n	A		5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6uip	C		4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	5a3x	D		n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	B	A	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	B	B	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	D	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	A	B	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	B	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6eif	A		4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1h	A	B	~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	C	B	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	C	B	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	7akb	A	B	4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	5a54	D		n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	A	A	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	D	B	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	4nct	B		pkc412	Human	Show
	DYRK1A	DYRK	CMGC	6eij	C		~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	B	B	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	7ajy	A		4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	5a4t	B		n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4nct	D		pkc412	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	A	B	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	C	A	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7ajs	A	B	4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	A	B	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	C	B	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	A	A	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	A	A	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	A	B	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a3x	B		n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7akb	A	A	4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	B	B	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7a4w	A		6-(4-methoxyphenyl)pyrimidine-2,4-diamine	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	B	B	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	5aik	C		4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj2	A	A	4-(4-methoxyphenyl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	B	B	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	4yll	A	B	10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	D	A	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	6a1f	A	A	8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	6ej4	B		3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline	Human	Show
	DYRK1A	DYRK	CMGC	5a4l	D	A	n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7fhs	A	A	(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	6s11	A	B	6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	A	A	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	3anq	C		(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	C	B	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	4aze	A		5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one	Human	Show
	DYRK1A	DYRK	CMGC	6s1b	A	B	~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	4yll	A	C	10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	6eiq	C		[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone	Human	Show
	DYRK1A	DYRK	CMGC	5a4t	D		n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7a53	A	A	(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	D	B	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	4mq1	C	A	n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6s1i	B	A	~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6ej4	C		3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline	Human	Show
	DYRK1A	DYRK	CMGC	2wo6	B	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	7a5b	A		4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	5a54	C		n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	A	B	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	A	A	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	6yf8	A		~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7o7k	A	A	n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	3anq	B		(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one	Human	Show
	DYRK1A	DYRK	CMGC	6eif	C		4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide	Human	Show
	DYRK1A	DYRK	CMGC	6eij	A		~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide	Human	Show
	DYRK1A	DYRK	CMGC	6yf8	C		~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	D	A	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	5a4e	C	B	n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	6s14	A	B	~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6eiv	C		~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	3anq	A		(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	B	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	B	A	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	7aja	A	A	1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine	Human	Show
	DYRK1A	DYRK	CMGC	4ylk	A	A	10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	4ylj	D	B	10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	7fht	A	A	(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	6eif	B		4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide	Human	Show
	DYRK1A	DYRK	CMGC	6s14	A	A	~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6uwy	D	B	4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide	Human	Show
	DYRK1A	DYRK	CMGC	4yu2	B	B	(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile	Human	Show
	DYRK1A	DYRK	CMGC	6eis	D	A	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	6t6a	B	A	4-chloranyl-5~{h}-cyclohepta[b]indol-10-one	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	D	B	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	5a54	B		n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	2wo6	B	B	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	7ajw	A	B	4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	7ajw	A	A	4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine	Human	Show
	DYRK1A	DYRK	CMGC	7fht	A	B	(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	6eij	D		~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide	Human	Show
	DYRK1A	DYRK	CMGC	7a5n	A		5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	B	A	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	7a5l	A	B	4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	7aj4	A	B	4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine	Human	Show
	DYRK1A	DYRK	CMGC	6eis	A	A	1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one	Human	Show
	DYRK1A	DYRK	CMGC	2vx3	D	A	n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide	Human	Show
	DYRK1A	DYRK	CMGC	6eir	D		~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide	Human	Show
	DYRK1A	DYRK	CMGC	6qu2	A	B	8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one	Human	Show
	DYRK1A	DYRK	CMGC	4yll	A	A	10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid	Human	Show
	DYRK1A	DYRK	CMGC	4mq2	A	B	methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate	Human	Show
	DYRK1A	DYRK	CMGC	7a4r	A	A	2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one	Human	Show
	DYRK1A	DYRK	CMGC	5a4q	D		n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide	Human	Show
	DYRK1A	DYRK	CMGC	7a4z	A		3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine	Human	Show

Division of Medicinal Chemistry - Vrije Universiteit Amsterdam