PDB-code
Search results (232 entries covering 121 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | B | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | Show |  |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | A | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | B | 4-methylbenzamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p79 | A | 1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylurea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | A | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | A | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | A | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | A | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | A | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | B | 1-phenylmethoxyurea | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | B | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | A | 6-methoxypyridine-3-carbothioamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | B | 2-phenoxyacetamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | A | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | A | 1-phenylmethoxyurea | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | B | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 1yw2 | A | 2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-one | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | A | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | B | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | A | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7c | A | 1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtm | A | 8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diium | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | A | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7z9t | A | n-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamide | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | B | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | B | thiophene-2-carbothioamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | B | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | B | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | B | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 8efj | A | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3py3 | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | B | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | A | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghl | A | 3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | B | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | B | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 8acm | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | A | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | A | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | B | benzyl hydroxycarbamate | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7a | A | 1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylurea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | A | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5o90 | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 4ka3 | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | B | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5uoj | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | A | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | B | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | B | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7be4 | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtn | A | 2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amine | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 7be5 | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamide | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | B | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p5k | A | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | A | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | B | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p4k | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2puu | A | 5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-ium | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | B | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 1lew | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | A | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | B | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | B | 6-methoxypyridine-3-carbothioamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | B | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2oza | B | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | A | benzyl hydroxycarbamate | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7b | A | 1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | A | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 1lez | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | A | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | A | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3p78 | A | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylurea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | A | 4-methylbenzamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghm | A | 3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | A | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | B | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | B | phosphothiophosphoric acid-adenylate ester | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | A | thiophene-2-carbothioamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 3tg1 | A | - | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | A | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdq | A | ~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamide | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | B | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | B | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | A | 2-phenoxyacetamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | B | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 1ywr | A | 4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-one | Mouse | Show | | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | A | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | A | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | B | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | A | - | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | |
