PDB-code
Browse kinase entries (page 127 of 282)
First 123 124 125 PreviousLast131 130 129 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | FGFR4 | FGFR | TK | 6nvj | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamide | Human | Show |  | |
| FGFR4 | FGFR | TK | 6nvk | A | A | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | Show | |
| FGFR4 | FGFR | TK | 6nvk | A | B | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | Show | |
| FGFR4 | FGFR | TK | 6v9c | A | A | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | Show | |
| FGFR4 | FGFR | TK | 6v9c | A | B | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | Show | |
| FGFR4 | FGFR | TK | 6yi8 | A | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | Show | |
| FGFR4 | FGFR | TK | 6yi8 | A | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | Show | |
| FGFR4 | FGFR | TK | 6yi8 | B | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | Show | |
| FGFR4 | FGFR | TK | 6yi8 | B | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | Show | |
| FGFR4 | FGFR | TK | 7dtz | A | n-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7f3m | A | 6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-one | Human | Show | | |
| FGFR4 | FGFR | TK | 7v29 | A | n-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7vjl | A | n-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7wct | A | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7wcw | A | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7wcx | A | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7ybo | A | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7ybp | A | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7ybx | A | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7yc1 | A | ~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 7yc3 | A | 6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | Show | | |
| FGFR4 | FGFR | TK | 8kh6 | A | - | Human | Show | | |
| FGFR4 | FGFR | TK | 8kh7 | A | - | Human | Show | | |
| FGFR4 | FGFR | TK | 8kh8 | A | - | Human | Show | | |
| FGFR4 | FGFR | TK | 8kh9 | A | - | Human | Show | | |
| FGFR4 | FGFR | TK | 8w5c | A | - | Human | Show | | |
| FGR | Src | TK | 7uy0 | A | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy0 | A | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy0 | A | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy0 | B | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy0 | B | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy0 | B | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
| FGR | Src | TK | 7uy3 | A | 3-[(6,7-dimethoxyquinazolin-4-yl)oxy]-n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methylbenzamide | Human | Show | | |
| FLT1 | VEGFR | TK | 3hng | A | A | n-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamide | Human | Show | |
| FLT1 | VEGFR | TK | 3hng | A | B | n-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamide | Human | Show | |
| FLT3 | PDGFR | TK | 1rjb | A | - | Human | Show | | |
| FLT3 | PDGFR | TK | 4rt7 | A | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | Show | |
| FLT3 | PDGFR | TK | 4rt7 | A | B | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | Show | |
| FLT3 | PDGFR | TK | 4xuf | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | Show | | |
| FLT3 | PDGFR | TK | 4xuf | B | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | Show | | |
| FLT3 | PDGFR | TK | 5x02 | A | n-[(2s)-1-[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxidanylidene-propan-2-yl]-4-(dimethylamino)-n-methyl-but-2-enamide | Human | Show | | |
| FLT3 | PDGFR | TK | 6il3 | A | A | 7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridine | Human | Show | |
| FLT3 | PDGFR | TK | 6il3 | A | B | 7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridine | Human | Show | |
| FLT3 | PDGFR | TK | 6jqr | A | 6-ethyl-3-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide | Human | Show | | |
| FYN | Src | TK | 2dq7 | X | staurosporine | Human | Show | | |
| GAK | NAK | Other | 4c57 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4c57 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4c57 | B | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4c57 | B | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | |
| GAK | NAK | Other | 4c58 | A | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | |
