PDB-code
Browse kinase entries (page 166 of 282)
First 162 163 164 PreviousLast170 169 168 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAP2K6 | STE7 | STE | 8p7j | A | n-[3-(1h-pyrrolo[2,3-b]pyridin-4-yl)phenyl]prop-2-enamide | Human | Show | ![]() | |
![]() | MAP2K6 | STE7 | STE | 8pm3 | A | ~{n}-[3-(2-azanylpyridin-4-yl)phenyl]propanamide | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 2dyl | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 3wzu | A | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 5b2k | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 5b2l | A | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 5b2l | A | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 5b2m | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 5y8u | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 5y90 | A | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 5y90 | A | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 5z1d | A | n-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamide | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 5z1e | A | n-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamide | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6ib0 | A | 1-[(3~{r})-3-(4-azanyl-3-ethynyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]prop-2-en-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6ib2 | A | 1-[(3~{r})-3-[4-azanyl-3-[1-(4-ethanoylphenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qfl | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qfr | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qft | A | 1-[(3~{r})-3-(4-azanyl-3-iodanyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qg4 | A | 1-[(3~{r})-3-[4-azanyl-3-(4-hydroxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qg7 | A | (r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qho | A | 1-[(3~{r})-3-(4-azanylpyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6qhr | A | 1-[(3~{r})-3-[4-azanyl-3-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6yfz | A | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yfz | A | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg0 | A | - | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6yg1 | A | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg1 | A | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg1 | B | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg1 | B | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg1 | C | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg1 | C | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg2 | A | A | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg2 | A | B | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg3 | A | A | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg3 | A | B | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg4 | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6yg5 | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile | Human | Show | ![]() | |
![]() | MAP2K7 | STE7 | STE | 6yg6 | A | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg6 | A | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg6 | B | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg6 | B | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg7 | A | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg7 | A | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg7 | B | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yg7 | B | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yz4 | A | A | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 6yz4 | A | B | - | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 7cbx | A | A | 3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 7cbx | A | B | 3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamide | Human | Show | ![]() |
![]() | MAP2K7 | STE7 | STE | 7ovi | A | 1-[(3~{r})-3-[4-azanyl-3-[1-(2-phenylethyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | ![]() |


