PDB-code
Browse kinase entries (page 191 of 282)
First 187 188 189 PreviousLast195 194 193 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK14 (p38a) | MAPK | CMGC | 3oc1 | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show |  | |
| MAPK14 (p38a) | MAPK | CMGC | 3ocg | A | 5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3od6 | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ody | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3odz | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | A | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | B | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3que | A | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3rin | A | n-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3roc | A | 3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3s3i | A | 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3s4q | A | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3u8w | A | 3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | A | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | B | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | A | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | B | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | A | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | B | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | B | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | B | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | A | 2-amino-phenylamino-dibenzosuberone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | B | 2-amino-phenylamino-dibenzosuberone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4a9y | A | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | B | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa4 | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa5 | A | n-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4aac | A | n-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4dli | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4dlj | A | 2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5b | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6a | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6c | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e8a | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh2 | A | 3-phenylquinazolin-4(3h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh3 | A | naringenin | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh4 | A | phenyl(piperidin-1-yl)methanone | Human | Show | |
