Browse kinase entries (page 241 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PRKCQ (PKCt)PKCAGC4ra5AB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHumanShow
PRKCQ (PKCt)PKCAGC4ra5BA(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHumanShow
PRKCQ (PKCt)PKCAGC4ra5BB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHumanShow
PRKCQ (PKCt)PKCAGC5f9eAA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHumanShow
PRKCQ (PKCt)PKCAGC5f9eAB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHumanShow
PRKCQ (PKCt)PKCAGC5f9eBA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHumanShow
PRKCQ (PKCt)PKCAGC5f9eBB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHumanShow
PRKG1 (PKG1)PKGAGC6bdlAA-HumanShow
PRKG1 (PKG1)PKGAGC6bdlAB-HumanShow
PRKG1 (PKG1)PKGAGC6bdlBA-HumanShow
PRKG1 (PKG1)PKGAGC6bdlBB-HumanShow
PRKG1 (PKG1)PKGAGC6bg2AAphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2ABphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2BAphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2BBphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2CAphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2CBphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2DAphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6bg2DBphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC6c0tAn-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamideHumanShow
PRKG1 (PKG1)PKGAGC7lv3Aphosphoaminophosphonic acid-adenylate esterHumanShow
PRKG1 (PKG1)PKGAGC7t4tAAadenosine-5'-triphosphateHumanShow
PRKG1 (PKG1)PKGAGC7t4tABadenosine-5'-triphosphateHumanShow
PRKG1 (PKG1)PKGAGC7t4uAA-HumanShow
PRKG1 (PKG1)PKGAGC7t4uAB-HumanShow
PRKG1 (PKG1)PKGAGC7t4vAA-HumanShow
PRKG1 (PKG1)PKGAGC7t4vAB-HumanShow
PRKG1 (PKG1)PKGAGC7t4wAA-HumanShow
PRKG1 (PKG1)PKGAGC7t4wAB-HumanShow
PRPF4B (PRP4)DYRKCMGC4ianA-HumanShow
PRPF4B (PRP4)DYRKCMGC4ianB-HumanShow
PRPF4B (PRP4)DYRKCMGC4ifcAAadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcABadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcBAadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcBBadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4iirAAphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4iirABphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4iirBAphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4iirBBphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpAA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpAB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpBA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpBB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6cnhAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6cnhAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjAA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjAB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjBA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjBB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjCA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
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