Search results (57 entries covering 35 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAP2K7STE7STE5y90AB-HumanShow
MAP2K7STE7STE5b2lAA-HumanShow
MAP2K7STE7STE5b2lAB-HumanShow
MAP2K7STE7STE6qflA-HumanShow
MAP2K7STE7STE6yg1AB-HumanShow
MAP2K7STE7STE6yg3AAn-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamideHumanShow
MAP2K7STE7STE5z1eAn-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamideHumanShow
MAP2K7STE7STE6qhrA1-[(3~{r})-3-[4-azanyl-3-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yg7BA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE6yz4AA-HumanShow
MAP2K7STE7STE7ovjAB1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yfzAB-HumanShow
MAP2K7STE7STE6qg7A(r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-oneHumanShow
MAP2K7STE7STE6qftA1-[(3~{r})-3-(4-azanyl-3-iodanyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yg1BA-HumanShow
MAP2K7STE7STE6yg1AA-HumanShow
MAP2K7STE7STE7ovkA1-[(3~{r})-3-[4-azanyl-3-[1-(5-bromanyl-2-oxidanyl-phenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yg7BB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE7ovnAB3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE6yg6BA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE6yg7AA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE6yg2AB1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yg6AB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE7ovnAA3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE7ovmAA~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE7cbxAA3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamideHumanShow
MAP2K7STE7STE6yg7AB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE6yg2AA1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE7cbxAB3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamideHumanShow
MAP2K7STE7STE6yfzAA-HumanShow
MAP2K7STE7STE6yg1BB-HumanShow
MAP2K7STE7STE6yg3ABn-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamideHumanShow
MAP2K7STE7STE5b2mA-HumanShow
MAP2K7STE7STE6qg4A1-[(3~{r})-3-[4-azanyl-3-(4-hydroxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6qfrA-HumanShow
MAP2K7STE7STE5y90AA-HumanShow
MAP2K7STE7STE2dylA-HumanShow
MAP2K7STE7STE7oviA1-[(3~{r})-3-[4-azanyl-3-[1-(2-phenylethyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE7ovmAB~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE3wzuA(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHumanShow
MAP2K7STE7STE6ib0A1-[(3~{r})-3-(4-azanyl-3-ethynyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]prop-2-en-1-oneHumanShow
MAP2K7STE7STE5b2kA-HumanShow
MAP2K7STE7STE6yg1CB-HumanShow
MAP2K7STE7STE6yg1CA-HumanShow
MAP2K7STE7STE6yg4A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHumanShow
MAP2K7STE7STE6yg6BB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE7ovlAB3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE6yg0A-HumanShow
MAP2K7STE7STE5z1dAn-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamideHumanShow
MAP2K7STE7STE7ovjAA1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6qhoA1-[(3~{r})-3-(4-azanylpyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE7ovlAA3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHumanShow
MAP2K7STE7STE6ib2A1-[(3~{r})-3-[4-azanyl-3-[1-(4-ethanoylphenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHumanShow
MAP2K7STE7STE6yg5A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrileHumanShow
MAP2K7STE7STE6yz4AB-HumanShow
MAP2K7STE7STE6yg6AA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHumanShow
MAP2K7STE7STE5y8uA-HumanShow