PDB-code
Browse kinase entries (page 111 of 282)
First 107 108 109 PreviousLast115 114 113 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | EIF2AK4 (GCN2) | PEK | Other | 7qwk | A | (2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamide | Human | Show |  | |
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | A | - | Human | Show | |
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | B | - | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 4p2k | A | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | A | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | B | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 4trl | A | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | A | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | B | - | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | A | - | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | B | - | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | A | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | B | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | A | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | B | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | A | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | B | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | A | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | B | alisertib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia1 | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | Show | | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | A | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | B | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | A | golvatinib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | B | golvatinib | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | A | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | B | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | A | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | B | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | B | - | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | C | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHA2 (EphA2) | Eph | TK | 5nk4 | A | A | 2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | Show | |
