Browse kinase entries (page 181 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAPK10 (JNK3)MAPKCMGC4x21Bn-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC4y46A1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylureaHumanShow
MAPK10 (JNK3)MAPKCMGC4y5hA1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylureaHumanShow
MAPK10 (JNK3)MAPKCMGC4z9lAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC4z9lABphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC6ekdAA4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6ekdAB4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhAA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhAB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhBA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhBB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhCA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhCB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhDA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6emhDB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC6eq9AAphosphomethylphosphonic acid adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC6eq9ABphosphomethylphosphonic acid adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC6eq9BAphosphomethylphosphonic acid adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC6eq9BBphosphomethylphosphonic acid adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC7ksiA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC7ksjA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC7kskA4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC7oreAA4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHumanShow
MAPK10 (JNK3)MAPKCMGC7oreAB4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHumanShow
MAPK10 (JNK3)MAPKCMGC7oreAC4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHumanShow
MAPK10 (JNK3)MAPKCMGC7orfAAn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC7orfABn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC7s1nAA4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC7s1nAB4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC7yl1A7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dioneHumanShow
MAPK10 (JNK3)MAPKCMGC8bzpAA2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHumanShow
MAPK10 (JNK3)MAPKCMGC8bzpAB2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHumanShow
MAPK10 (JNK3)MAPKCMGC8enjAn-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamideHumanShow
MAPK10 (JNK3)MAPKCMGC8wgfAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK10 (JNK3)MAPKCMGC8wgfABphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK11 (p38b)MAPKCMGC3gc8A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHumanShow
MAPK11 (p38b)MAPKCMGC3gc8B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHumanShow
MAPK11 (p38b)MAPKCMGC3gc9A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHumanShow
MAPK11 (p38b)MAPKCMGC3gc9B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHumanShow
MAPK11 (p38b)MAPKCMGC3gp0AAnilotinibHumanShow
MAPK11 (p38b)MAPKCMGC3gp0ABnilotinibHumanShow
MAPK11 (p38b)MAPKCMGC8ygwA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHumanShow
MAPK12 (p38g)MAPKCMGC1cm8Aphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK12 (p38g)MAPKCMGC1cm8Bphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK12 (p38g)MAPKCMGC6unaAA-HumanShow
MAPK12 (p38g)MAPKCMGC6unaAB-HumanShow
MAPK12 (p38g)MAPKCMGC6unaBA-HumanShow
MAPK12 (p38g)MAPKCMGC6unaBB-HumanShow
MAPK12 (p38g)MAPKCMGC7cgaA-HumanShow
MAPK13 (p38d)MAPKCMGC3coiAA-HumanShow
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