PDB-code
Browse kinase entries (page 181 of 282)
First 177 178 179 PreviousLast185 184 183 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4x21 | B | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4y46 | A | 1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylurea | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4y5h | A | 1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylurea | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | A | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | B | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ksi | A | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ksj | A | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ksk | A | 4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | A | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | B | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | C | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | A | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | B | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | A | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | B | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 7yl1 | A | 7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dione | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | A | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | B | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 8enj | A | n-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gc8 | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gc8 | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gc9 | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gc9 | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | ![]() | |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | A | nilotinib | Human | Show | ![]() |
![]() | MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | B | nilotinib | Human | Show | ![]() |
![]() | MAPK11 (p38b) | MAPK | CMGC | 8ygw | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | ![]() | |
![]() | MAPK12 (p38g) | MAPK | CMGC | 1cm8 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK12 (p38g) | MAPK | CMGC | 1cm8 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK12 (p38g) | MAPK | CMGC | 6una | A | A | - | Human | Show | ![]() |
![]() | MAPK12 (p38g) | MAPK | CMGC | 6una | A | B | - | Human | Show | ![]() |
![]() | MAPK12 (p38g) | MAPK | CMGC | 6una | B | A | - | Human | Show | ![]() |
![]() | MAPK12 (p38g) | MAPK | CMGC | 6una | B | B | - | Human | Show | ![]() |
![]() | MAPK12 (p38g) | MAPK | CMGC | 7cga | A | - | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 3coi | A | A | - | Human | Show | ![]() |


