PDB-code
Browse kinase entries (page 197 of 282)
First 193 194 195 PreviousLast201 200 199 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2jbp | L | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2onl | C | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2onl | D | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2oza | A | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2p3g | X | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2pzy | A | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2pzy | B | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2pzy | C | staurosporine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 2pzy | D | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | A | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | B | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | C | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | D | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | E | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | F | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | G | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | H | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | I | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | J | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | K | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3a2c | L | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3fpm | A | 3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3fyj | X | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3fyk | X | (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | C | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | D | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | E | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | F | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | G | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | H | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | I | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | J | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | K | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3gok | L | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3ka0 | A | 6-{5-[(2-aminopyrimidin-4-yl)amino]-2-hydroxyphenyl}-n-methylidene-1-benzothiophene-2-carboxamide | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | A | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | B | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | C | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | D | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | E | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | F | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | G | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | H | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | I | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | J | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | K | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | L | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | A | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | Show | ![]() |


