PDB-code
Browse kinase entries (page 198 of 282)
First 194 195 196 PreviousLast202 201 200 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | B | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | A | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | B | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3m42 | A | 2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7h-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | A | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | B | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | C | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | D | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | E | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | F | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | G | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | H | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | I | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | J | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | K | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2b | L | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r2y | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | A | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | B | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | A | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | B | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | C | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | D | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | E | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | F | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | B | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6t8x | A | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | B | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | B | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | B | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | B | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 8xu4 | A | - | Human | Show | ![]() | |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | A | - | Human | Show | ![]() |
![]() | MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | B | - | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | A | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | B | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | A | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | B | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3she | A | A | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 3she | A | B | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | MARK1 | CAMKL | CAMK | 2hak | A | - | Human | Show | ![]() |


