Browse kinase entries (page 215 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PAK4STE20STE8yhkA-HumanShow
PAK5STE20STE2f57AA-HumanShow
PAK5STE20STE2f57AB-HumanShow
PAK5STE20STE2f57BAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHumanShow
PAK5STE20STE2f57BBn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHumanShow
PAK5STE20STE8c12AA-HumanShow
PAK5STE20STE8c12AB-HumanShow
PAK6STE20STE2c30AA-HumanShow
PAK6STE20STE2c30AB-HumanShow
PAK6STE20STE4ks7AApf-3758309HumanShow
PAK6STE20STE4ks7ABpf-3758309HumanShow
PAK6STE20STE4ks8AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHumanShow
PAK6STE20STE4ks8ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHumanShow
PASKCAMKLCAMK3dlsAadenosine-5'-diphosphateHumanShow
PASKCAMKLCAMK3dlsBadenosine-5'-diphosphateHumanShow
PASKCAMKLCAMK3dlsCadenosine-5'-diphosphateHumanShow
PASKCAMKLCAMK3dlsDadenosine-5'-diphosphateHumanShow
PASKCAMKLCAMK3dlsEadenosine-5'-diphosphateHumanShow
PASKCAMKLCAMK3dlsFadenosine-5'-diphosphateHumanShow
PBKTOPKOther5j0aA-HumanShow
PBKTOPKOther5j0aB-HumanShow
PDGFRA (PDGFRa)PDGFRTK5grnAAn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHumanShow
PDGFRA (PDGFRa)PDGFRTK5grnABn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHumanShow
PDGFRA (PDGFRa)PDGFRTK5k5xA-HumanShow
PDGFRA (PDGFRa)PDGFRTK6a32A-HumanShow
PDGFRA (PDGFRa)PDGFRTK6joiA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHumanShow
PDGFRA (PDGFRa)PDGFRTK6jojA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHumanShow
PDGFRA (PDGFRa)PDGFRTK6jokAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHumanShow
PDGFRA (PDGFRa)PDGFRTK6jolA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHumanShow
PDGFRA (PDGFRa)PDGFRTK8pqhA(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHumanShow
PDGFRA (PDGFRa)PDGFRTK8pqiAA(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHumanShow
PDGFRA (PDGFRa)PDGFRTK8pqiAB(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHumanShow
PDGFRA (PDGFRa)PDGFRTK8pqjAA-HumanShow
PDGFRA (PDGFRa)PDGFRTK8pqjAB-HumanShow
PDGFRA (PDGFRa)PDGFRTK8pqkAA-HumanShow
PDGFRA (PDGFRa)PDGFRTK8pqkAB-HumanShow
PDPK1 (PDK1)PDK1AGC1h1wAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC1h1wABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC1okyAAstaurosporineHumanShow
PDPK1 (PDK1)PDK1AGC1okyABstaurosporineHumanShow
PDPK1 (PDK1)PDK1AGC1okzA7-hydroxystaurosporineHumanShow
PDPK1 (PDK1)PDK1AGC1uu3AA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu3AB(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu7A3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu8AA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu8AB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu9AA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uu9AB3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1uvrA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHumanShow
PDPK1 (PDK1)PDK1AGC1z5mAn-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)amino]phenyl}amino)pyrimidin-4-yl]amino}propyl)-2,2-dimethylmalonamideHumanShow
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